Tag: Modulator|Activator

For research use only. We do not sell to patients. Idebenone CAS No. : 58186-27-9 Biological Activity：Idebenone, a well-appreciated mitochondrial protectant, exhibits protective efficacy against neurotoxicity and can be used for the research of Alzheimer’s disease, Huntington’s disease. Idebenone (oxidised form) has a dose-dependent inhibitory effect on the enzymatic metabolism of arachidonic acid in astroglial […]

For research use only. We do not sell to patients. Clobenpropit dihydrobromide CAS No. : 145231-35-2 Biological Activity：Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors […]

For research use only. We do not sell to patients. Uridine 5′-diphosphate sodium salt CAS No. : 21931-53-3 Biological Activity：Uridine 5′-diphosphate sodium salt is a potent, selective P2Y6 receptor native agonist (EC50=300 nM; pEC50=6.52) and a potent P2Y14 antagonist (pEC50=7.28). Uridine 5′-diphosphate sodium salt, an endogenous metabolite, catalyzes the glucuronidation of a wide array of […]

For research use only. We do not sell to patients. Uridine-5′-diphosphate disodium salt CAS No. : 27821-45-0 Biological Activity：Uridine-5′-diphosphate disodium salt is a potent, selective P2Y6 receptor native agonist (EC50=300 nM; pEC50=6.52 for human P2Y6 receptor). Uridine-5′-diphosphate disodium salt, an endogenous metabolite, catalyzes the glucuronidation of a wide array of substrates and is used in […]