Tag: Modulator

For research use only. We do not sell to patients. DL-Norepinephrine hydrochloride CAS No. : 55-27-6 Biological Activity：DL-Norepinephrine hydrochloride is a synthetic phenylethylamine that mimics the sympathomimetic actions of the endogenous norepinephrine．DL-Norepinephrine hydrochloride is a neurotransmitter targets α1 and β1 adrenoceptors, has an increasing effect on subendocardial oxygen tension. Research Area：Neurological Disease|Endocrinology Targets：Adrenergic Receptor Related […]

For research use only. We do not sell to patients. Cimetidine CAS No. : 51481-61-9 Biological Activity：Cimetidine (SKF-92334) is an orally active and inverse histamine H2 receptor antagonist with a Ki of 0.6 μM. Cimetidine is a gastric acid reducer, and can be used for duodenal and gastric ulcers research. Cimetidine has anti-cancer and anti-inflammatory […]

For research use only. We do not sell to patients. Bradykinin (1-7) CAS No. : 23815-87-4 Biological Activity：Bradykinin (1-7) is an amino-truncated Bradykinin peptide. Bradykinin (1-7) is a metabolite of Bradykinin, cleaved by endopeptidase. Research Area：Cardiovascular Disease|Endocrinology Targets：Bradykinin Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Cardiovascular Disease Compound Library;Endocrinology Compound Library;Neurotransmitter Receptor Compound […]

For research use only. We do not sell to patients. GLP-1R modulator L7-028 CAS No. : 2648317-95-5 Biological Activity：GLP-1R modulator L7-028 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 11.01 ± 2.73 μM). Research Area：Metabolic Disease Targets：GCGR Related Small Molecules:BETP;GLP-1R agonist 4;VU0453379;PF-06291874;Utreglutide;TT-OAD2;Efocipegtrutide;GLP-1 receptor agonist 2;NNC-0640;Cochinchinenin C;{Val1}-Exendin-3/4;GLP-1(28-36)amide TFA;Exendin-4 acetate;Glepaglutide;GLP-1(7-37);GLP-1 receptor […]

For research use only. We do not sell to patients. Fluorogen binding modulator-1 CAS No. : 510716-65-1 Biological Activity：Fluorogen binding modulator-1 (PubChem SID 125240934) is a fluorogen activating protein (FAP)-fluorogen binding modulator with -log EC50s of 6.61 and 6.37 for AM2.2-β2AR and AM2.2-GPR32, respectively. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl […]

For research use only. We do not sell to patients. P-gp modulator 2 Biological Activity：P-gp modulator 2 (Compound 27) is a potent, competitive, allosteric P-glycoprotein (P-gp) modulator. Research Area：Cancer Targets：P-glycoprotein Related Small Molecules:Biricodar;P-gp inhibitor 4;Sinapine thiocyanate;Dofequidar fumarate;Elacridar;Coniferyl ferulate;Anticancer agent 50;Valspodar;P-gp inhibitor 1;Boeravinone B;Solamargine;Polyoxyethylene stearate;TTT-28;CP-100356 hydrochloride;Epoxylathyrol;Chrysosplenetin;Zamicastat;Tariquidar;P-gp modulator 3;Roemerine;Coleon-U-quinone;Zosuquidar trihydrochloride;Encequidar;P-gp modulator 1 Trending products：Recombinant Proteins  |  Bioactive […]

For research use only. We do not sell to patients. Raloxifene CAS No. : 84449-90-1 Biological Activity：Raloxifene (Keoxifene) is a benzothiophene-derived selective estrogen receptor modulator (SERM). Raloxifene has estrogen-agonistic effects on bone and lipids and estrogen-antagonistic effects on the breast and uterus. Raloxifene is used for breast cancer and osteoporosis research. Research Area：Cancer Targets：Estrogen Receptor/ERR […]

For research use only. We do not sell to patients. Tracazolate hydrochloride CAS No. : 1135210-68-2 Biological Activity：Tracazolate (ICI 136753) hydrochloride is a potent GABAA receptor modulator. Tracazolate hydrochloride has selectivity for β3 and potentiates α1β1γ2s (EC50=13.2 μM), α1β3γ2 (EC50=1.5 μM). Tracazolate hydrochloride has the potency (EC50) determined by the nature of the third subunit […]

For research use only. We do not sell to patients. CFTR corrector 2 CAS No. : 1628416-28-3 Biological Activity：CFTR corrector 2 is a cystic fibrosis transmembrane conductance corrector (CFTR), extracted from patent US20140274933. Research Area：Inflammation/Immunology|Cancer Targets：CFTR|Autophagy Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Membrane Transporter/Ion Channel Compound Library;Anti-Cancer […]

For research use only. We do not sell to patients. Substance P (alligator) CAS No. : 113516-47-5 Biological Activity：Substance P (alligator), a Substance P (Substance P (HY-P0201)) extracted from alligator, is a neuropeptide. The primary structure of Substance P (alligator) is: Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2. Research Area：Neurological Disease Targets：Neurokinin Receptor|Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide N-oxide;3-Hydroxyglutaric acid-d5;DPPC-d62;SDMA-d6;2-Mercaptobenzothiazole;N-Acetyl-L-glutamic […]