Tag: Modulator

For research use only. We do not sell to patients. BMS453 CAS No. : 166977-43-1 Biological Activity：BMS453 (BMS-189453), a synthetic retinoid, is a RARβ agonist and a RARα/RARγ antagonist. BMS453 inhibits breast cell growth predominantly through the induction of active TGFβ[2]. Research Area：Cancer Targets：RAR/RXR Related Screening Libraries:Natural Product-like Compound Library;Bioactive Compound Library Plus;Metabolism/Protease Compound Library;Anti-Cancer […]

For research use only. We do not sell to patients. P-gp modulator 3 Biological Activity：P-gp modulator 3 (Compound 37) is a potent, competitive, allosteric P-glycoprotein (P-gp) modulator. Research Area：Cancer Targets：P-glycoprotein Related Small Molecules:Biricodar;P-gp inhibitor 4;Sinapine thiocyanate;Dofequidar fumarate;Elacridar;Coniferyl ferulate;Anticancer agent 50;Valspodar;P-gp inhibitor 1;Boeravinone B;Solamargine;Polyoxyethylene stearate;TTT-28;CP-100356 hydrochloride;Epoxylathyrol;Chrysosplenetin;Zamicastat;Tariquidar;Roemerine;Coleon-U-quinone;Zosuquidar trihydrochloride;Encequidar;P-gp modulator 1 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  […]

For research use only. We do not sell to patients. GP531 CAS No. : 142344-87-4 Biological Activity：GP531 is a potent, second-generation adenosine regulating agent, is pharmacologically silent under basal conditions but increases localized endogenous adenosine during ischemia. Research Area：Cardiovascular Disease Targets：Adenosine Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Small Molecule Immuno-Oncology Compound Library;Anti-Cardiovascular […]

For research use only. We do not sell to patients. Betahistine mesylate CAS No. : 54856-23-4 Biological Activity：Betahistine mesylate is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. Betahistine mesylate is used for the study of rheumatoid arthritis (RA)[3]. Research Area：Inflammation/Immunology Targets：Histamine Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug […]

For research use only. We do not sell to patients. Carbidopa CAS No. : 28860-95-9 Biological Activity：Carbidopa ((S)-(-)-Carbidopa), a peripheral decarboxylase inhibitor, can be used for the research of Parkinson’s disease. Carbidopa is a selective aryl hydrocarbon receptor (AhR) modulator. Carbidopa inhibits pancreatic cancer cell and tumor growth[2]. Research Area：Cancer|Neurological Disease Targets：Aryl Hydrocarbon Receptor Related […]

For research use only. We do not sell to patients. Ph-HTBA CAS No. : 2368927-41-5 Biological Activity：Ph-HTBA is a high-affinity, brain-penetrating modulator for CaMKIIα. Ph-HTBA has binding affinity for CaMKIIα with a Kd value of 757 nM. Ph-HTBA can be used for the research of ischemia and neurodegenerative disorders. Research Area：Neurological Disease Targets：CaMK Related Small […]

For research use only. We do not sell to patients. NEO 376 CAS No. : 496921-73-4 Biological Activity：NEO 376 is a selective modulator of 5-HT1 receptor, GABA receptor and dopamine receptor, with anti-psychotic actively. Research Area：Neurological Disease Targets：Dopamine Receptor|5-HT Receptor|GABA Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Membrane Transporter/Ion Channel Compound Library;Neuronal Signaling […]

For research use only. We do not sell to patients. AZD-6280 CAS No. : 942436-93-3 Biological Activity：AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. Research Area：Neurological Disease Targets：GABA Receptor Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus; Related Small Molecules:SKF89976A hydrochloride;mGAT-IN-1;Alpidem;FG8119;Valerenic acid;Picrotoxinin;Miltirone;Etifoxine-13C,d3;Adipiplon;Gabazine;Broflanilide;Fluxametamide;ONO-8590580;γ-Aminobutyric acid-d6;Ginsenoside Rc;Fipronil;p-Hydroxybenzaldehyde-13C;Lesogaberan hydrochloride;FG 7142;Isoguvacine hydrochloride;Guvacine ethyl […]

For research use only. We do not sell to patients. Triamcinolone Benetonide CAS No. : 31002-79-6 Biological Activity：Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity. Research Area：Inflammation/Immunology|Endocrinology Targets：Glucocorticoid Receptor Related Small Molecules:Deflazacort-D5;PPARγ/GR modulator 1;Glucocorticoid receptor agonist-2;AZD2906;Beclometasone dipropionate;ORIC-101;Clobetasone butyrate;Cortisone-d2;Clobetasone butyrate-d7;Cortisone-13C3;Glucocorticoid receptor agonist;Cortodoxone-d2;Hydrocortisone aceponate;Glucocorticoid receptor-IN-2;OP-3633;GW-870086;Nenocorilant;Hydrocortisone cypionate;Corticosterone-d8;21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione;Deflazacort-d5-1;Mapracorat;Hydrocortisone-d4;Hydrocortisone acetate Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  […]

For research use only. We do not sell to patients. Myomodulin CAS No. : 110570-93-9 Biological Activity：Myomodulin is a neuropeptide present in molluscs, insects, and gastropods. Research Area：Neurological Disease Targets：Calcium Channel|Sodium Channel|Potassium Channel Related Small Molecules:Benidipine hydrochloride;Lu AE98134;CaV1.3 antagonist-1;14-Deoxyandrographolide;Kv3 modulator 2;Zandatrigine;(Rac)-MEM 1003;Glaucine;Veratridine;Efonidipine hydrochloride monoethanolate;L-Ascorbic acid sodium salt;Brompheniramine-d6 maleate;Pinacidil;MRS 1523;GX-674;Nilvadipine;AMP-PNP tetralithium;Dibucaine;IK1 inhibitor PA-6;Lercanidipine;CP-060;VU590;Sodium Channel inhibitor 2 […]