Tag: inhibitor

For research use only. We do not sell to patients. PKI 14-22 amide,myristoylated TFA Biological Activity：PKI 14-22 amide,myristoylated TFA is a potent cAMP-dependent PKA inhibitor. PKI 14-22 amide,myristoylated TFA reduces the IgG-mediated phagocytic response and also inhibits neutrophil adhesion. Research Area：Cancer Targets：PKA Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:Staurosporine;Malantide;DS89002333;Rp-8-CPT-cAMPS sodium;PF-4950834;Warangalone;STAD 2;AT13148;CCG215022;KT5720;8-Bromo-cAMP sodium […]

For research use only. We do not sell to patients. Ibrutinib dimer CAS No. : 2031255-23-7 Biological Activity：Ibrutinib dimer is a Dimer of Ibrutinib. Ibrutinib dimer is an impurity of Ibrutinib. Ibrutinib is a selective, irreversible Btk inhibitor with an IC50 of 0.5 nM[2]. Research Area：Cancer Targets：Btk Related Small Molecules:JAK3/BTK-IN-1;Elsubrutinib;ARQ 531;PF-06250112;PCI 29732;CHMFL-EGFR-202;Avitinib;RN486;GDC-0834 Racemate;Spebrutinib besylate;Vecabrutinib;BMX-IN-1;Tolebrutinib;BTK-IN-16;(R)-Zanubrutinib;Pirtobrutinib;CTA056;EGFR-IN-40;QL-X-138;ACP-5862;BTK-IN-12;JAK3/BTK-IN-4;JAK3/BTK-IN-6;BTK inhibitor […]

For research use only. We do not sell to patients. Lenampicillin hydrochloride CAS No. : 80734-02-7 Biological Activity：Lenampicillin hydrochloride (KBT 1585 hydrochloride) is an orally active prodrug of Ampicillin and is an effective beta-lactam antibacterial agent that inhibits bacterial penicillin-binding proteins (transpeptidase). Lenampicillin hydrochloride has improved absorption and decreased side effects compares to Ampicillin and […]

For research use only. We do not sell to patients. Antibacterial agent 45 CAS No. : 1426572-50-0 Biological Activity：Antibacterial agent 45, an antibacterial agent, significantly lowers MIC value of antibacterial agent Ceftazidime. Research Area：Infection Targets：Bacterial Related Small Molecules:Sandramycin;LLO (91-99);Gepotidacin;Oritavancin;Azlocillin sodium salt;Herbimycin A;Leucomycin;Isouvaretin;Antibacterial agent 99;Nafcillin;Antitubercular agent-28;Ochromycinone;Staurosporine;Nucleocidin;(±)-Leucine-13C-1;Ciclopirox-d11;Ciclopirox olamine;Clotrimazole-d5;SQ109;Neomycin sulfate;Bauer-7-ene-3β,16α-diol;Aminothiazole Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  […]

For research use only. We do not sell to patients. ATX inhibitor 22 Biological Activity：ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) with IC50 of 218 nM but lost its inhibitory activity of LPAR1. Research Area：Cancer Targets：Phosphodiesterase (PDE) Related Small Molecules:Senazodan hydrochloride;(E/Z)-HA155;Enpp/Carbonic anhydrase-IN-1;Carbazeran citrate;Bay 60-7550;BC11-38;Deltarasin hydrochloride;Glaucine;Ziritaxestat;Udenafil-d7;D159687;ITI-214;PDE10-IN-5;ICI 153110;Furamidine dihydrochloride;ML-030;PDE4-IN-10;Mirodenafil-d7 dihydrochloride;PDE1-IN-4;PDE4B-IN-3;Cirsimarin;PF-03049423;IBMX;Pimobendan;Gisadenafil besylate;S32826 disodium Trending products：Recombinant […]

For research use only. We do not sell to patients. Debneyol CAS No. : 99694-82-3 Biological Activity：Debneyol exhibits more potent fungicidal activity than validamycin. Research Area：Infection Targets：Fungal Related Small Molecules:Antifungal agent 20;Haloprogin;Staurosporine;Ciclopirox-d11;Ciclopirox olamine;Clotrimazole-d5;(R)-Camptothecin-d5;Ticlatone;Aminothiazole;Magnesium silicate;α-Terpinene;Hydroxyphenyllactic acid;Iprobenfos;Chlorphenesin;Moniliformin sodium salt;HLF1-11;β-Amyrin acetate;Bifonazole;Aszonapyrone A;Oenothein B;Pyrimorph;(+)-Magnoflorine iodide;Antifungal agent 39 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent […]

For research use only. We do not sell to patients. NSC81111 CAS No. : 1678-14-4 Biological Activity：NSC81111 is a potent and orally active EGFR-TK inhibitor with an IC50 of 0.15 nM. NSC81111 has anticaner effects. Research Area：Cancer Targets：EGFR Related Small Molecules:pp60 (v-SRC) Autophosphorylation Site, Phosphorylated;BMS-690514;Osimertinib-13C,d3;EGFR-IN-5;FGFR2-IN-3;Genistein;Epertinib hydrochloride;UNC-CA359;Osimertinib mesylate;AV-412 free base;Nelipepimut-S;Falnidamol;HER2-IN-6;PROTAC EGFR degrader 7;CHMFL-EGFR-202;Avitinib;Naquotinib;Lavendustin A;EAI001;EGFR/HER2/CDK9-IN-2;Cyasterone;DP-C-4;Allitinib Trending products：Recombinant […]

For research use only. We do not sell to patients. Leucomycin CAS No. : 1392-21-8 Biological Activity：Leucomycin (kitasamycin) is a macrolide antibiotic produced by Streptomyces kitasatoensis[2][3][4]. Research Area：Infection Targets：Bacterial|Antibiotic Related Screening Libraries:Natural Product Library Plus;Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Anti-Infection Compound Library;Natural Product Library;FDA-Approved Drug Library;Drug Repurposing […]

For research use only. We do not sell to patients. Nebicapone CAS No. : 274925-86-9 Biological Activity：Nebicapone (BIA 3-202), a reversible catechol-O-methyltransferase (COMT) inhibitor, is mainly metabolized by glucuronidation. Nebicapone is mainly peripherally acting inhibitor that decreases the biotransformation of L-DOPA to 3-O-methyl-DOPA by inhibition of COMT, and it is potential for the treatment of […]

For research use only. We do not sell to patients. Ametantrone CAS No. : 64862-96-0 Biological Activity：Ametantrone (NSC 196473) is an antitumor agent that intercalates into DNA and induces topoisomerase II (TOP2)-mediated DNA break. Research Area：Cancer Targets：DNA/RNA Synthesis Related Small Molecules:ddCTP trisodium;7-TFA-ap-7-Deaza-dA;P1788;Thymidine-13C5,15N;NSC 617145;116-9e;DNA Gyrase-IN-5;DMT-2′-F-Bz-dA;6-Thio-2′-Deoxyguanosine;Antitumor agent-74;Risdiplam;TH287 hydrochloride;Direct Black 38;7-TFA-ap-7-Deaza-ddA;BCH001;NKP-1339;Fialuridine;2′-O-MOE-5-Me-rC;PTC299;2′-F-Bz-dC Phosphoramidite Trending products：Recombinant Proteins  |  Bioactive Screening […]