Tag: inhibitor

For research use only. We do not sell to patients. Lenvatinib-d4 Biological Activity：Lenvatinib-d4 (E7080-d4) is the deuterium labeled Lenvatinib. Lenvatinib (E7080) is an oral, multi-targeted tyrosine kinase inhibitor that inhibits VEGFR1-3, FGFR1-4, PDGFR, KIT, and RET, shows potent antitumor activities[2]. Research Area：Cancer Targets：VEGFR|RET|c-Kit|FGFR|PDGFR Related Small Molecules:(Z)-FeCP-oxindole;VEGFR-2-IN-24;BMS-690514;PROTAC VEGFR-2 degrader-2;Henatinib;PI3K/VEGFR2-IN-1;c-Kit-IN-5-1;Flumatinib mesylate;IHMT-TRK-284;RET-IN-18;Ferulic acid-13C3;PDGFRα/FLT3-ITD-IN-2;FGFR-IN-7;PP58;Hydroxytanshinone IIA;Chiauranib;Foretinib;ZM323881 hydrochloride;Zeteletinib;FGFR3-IN-1;Pexidartinib;PTC299;ENMD-2076 Tartrate;Aflibercept Trending products：Recombinant […]

For research use only. We do not sell to patients. VI 16832 CAS No. : 1430218-51-1 Biological Activity：VI 16832 is a broad spectrum Type I kinase inhibitor which can be used as an enrichment tool for the comparative expression analysis of protein kinases in different cancer cell lines. Research Area：Cancer Targets：Others Related Screening Libraries:Bioactive Compound […]

For research use only. We do not sell to patients. 3-Fucosyllactose CAS No. : 41312-47-4 Biological Activity：3-Fucosyllactose (3-Fucosyl-D-lactose) is one of the major fucosylated oligosaccharides found in human breast milk. 3-Fucosyllactose shows prebiotic, immunomodulator, neonatal brain development, and antimicrobial function. Research Area：Infection|Inflammation/Immunology|Neurological Disease Targets：Enterovirus|Bacterial Related Small Molecules:Sandramycin;LLO (91-99);Gepotidacin;Oritavancin;Azlocillin sodium salt;Herbimycin A;Antibacterial agent 45;Leucomycin;Isouvaretin;Antibacterial agent 99;Nafcillin;Antitubercular […]

For research use only. We do not sell to patients. MNITMT CAS No. : 177653-76-8 Biological Activity：MNITMT is a more potent immunosuppressive agent without bone marrow toxicity. Research Area：Inflammation/Immunology Targets：Others Related Screening Libraries:Bioactive Compound Library Plus;Immunology/Inflammation Compound Library; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant […]

For research use only. We do not sell to patients. ELN318463 CAS No. : 851600-86-7 Biological Activity：ELN318463 is an amyloid precursor protein (APP) selective γ-secretase inhibitor. ELN318463 shows differential inhibition of presenilin (PS1)- and PS2-comprised γ-secretase with EC50s of 12 nM and 656 nM for PS1 and PS2, respectively. ELN318463 is 51-fold more selective for […]

For research use only. We do not sell to patients. Entacapone CAS No. : 130929-57-6 Biological Activity：Entacapone is a potent, reversible, peripherally acting and orally active catechol-O-methyltransferase (COMT) inhibitor. Entacapone inhibits COMT from rat brain, erythrocytes and liver with IC50 values of 10 nM, 20 nM, and 160 nM, respectively. Entacapone is selective for COMT […]

For research use only. We do not sell to patients. D-(-)-3-Phosphoglyceric acid disodium CAS No. : 80731-10-8 Biological Activity：D-(-)-3-Phosphoglyceric acid (3-Phospho-D-glyceric acid) disodium is an important intermediate in the enzyme-catalysed process of glycolysis. D-(-)-3-Phosphoglyceric acid disodium competitively inhibits yeast enolase[2]. Research Area：Infection Targets：Enolase Related Small Molecules:POMHEX;AP-III-a4 hydrochloride;SF2312 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  […]

For research use only. We do not sell to patients. D6808 Biological Activity：D6808 is a highly selective and potent c‑Met inhibitor with an IC50 value of 2.9 nM. D6808 induces cell apoptosis and cell cycle arrest. D6808 can be used for the research of NSCLC and gastric cancers. Research Area：Cancer Targets：c-Met/HGFR Related Small Molecules:AMG-208;MET kinase-IN-2;c-Met-IN-9;Tyrosine […]

For research use only. We do not sell to patients. USP7-IN-1 CAS No. : 1381291-36-6 Biological Activity：USP7-IN-1 is a selective and reversible inhibitor of ubiquitin-specific protease 7 (USP7), with an IC50 of 77 μM, and can be used for the research of cancer. Research Area：Cancer Targets：Deubiquitinase Related Screening Libraries:Bioactive Compound Library Plus;Cell Cycle/DNA Damage Compound […]

For research use only. We do not sell to patients. Herbimycin A CAS No. : 70563-58-5 Biological Activity：Herbimycin A, an ansamycin antibiotic, acts as a Src family kinase inhibitor. Herbimycin A binds to the SH domain and inhibits the activity of p60v-src and p210BCR-ABL Herbimycin A inhibits Hsp90 and impairs recovery from heat shock. Herbimycin […]