Tag: Inducer|Antagonist|Inhibitor

For research use only. We do not sell to patients. Mefloquine hydrochloride CAS No. : 51773-92-3 Biological Activity：Mefloquine hydrochloride (Mefloquin hydrochloride), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine hydrochloride is also a K+ channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine hydrochloride can be used for malaria, systemic lupus erythematosus […]

For research use only. We do not sell to patients. Fasudil Hydrochloride CAS No. : 105628-07-7 Biological Activity：Fasudil (HA-1077; AT877) Hydrochloride is a nonspecific RhoA/ROCK inhibitor and also has inhibitory effect on protein kinases, with an Ki of 0.33 μM for ROCK1, IC50s of 0.158 μM and 4.58 μM, 12.30 μM, 1.650 μM for ROCK2 […]

For research use only. We do not sell to patients. Mifepristone-13C,d3 Biological Activity：Mifepristone-13C,d3 is the 13C- and deuterium labeled Mifepristone. Mifepristone (RU486) is a progesterone receptor (PR) and glucocorticoid receptor (GR) antagonist with IC50s of 0.2 nM and 2.6 nM in in vitro assay. Research Area：Endocrinology|Cancer Targets：Autophagy|Glucocorticoid Receptor|Progesterone Receptor|NO Synthase Related Small Molecules:Carboxy-PTIO potassium;Valeriandoid F;Gestonorone […]