Tag: Inducer|Antagonist

For research use only. We do not sell to patients. Fulvestrant-d3 Biological Activity：Fulvestrant-d3 (ICI 182780-d3) is the deuterium labeled Fulvestrant. Fulvestrant (ICI 182780) is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC50 of 9.4 nM. Fulvestrant is also a GPR30 agonist. Fulvestrant effectively inhibits the growth of ER-positive MCF-7 cells […]

For research use only. We do not sell to patients. SM-164 Hydrochloride Biological Activity：SM-164 Hydrochloride is a cell-permeable Smac mimetic compound. SM-164 binds to XIAP protein containing both the BIR2 and BIR3 domains with an IC50 value of 1.39 nM and functions as an extremely potent antagonist of XIAP. Research Area：Cancer Targets：IAP|Apoptosis Related Screening Libraries:Bioactive […]

For research use only. We do not sell to patients. Degarelix CAS No. : 214766-78-6 Biological Activity：Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR/LHRHR) antagonist. Degarelix can be used for prostate cancer research. Research Area：Cancer|Endocrinology Targets：GnRH Receptor|Apoptosis Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Apoptosis […]

For research use only. We do not sell to patients. Cisatracurium besylate CAS No. : 96946-42-8 Biological Activity：Cisatracurium besylate (51W89) is a nondepolarizing neuromuscular blocking agent, antagonizing the action of acetylcholine by inhibiting neuromuscular transmission. Research Area：Neurological Disease|Cancer Targets：nAChR|Autophagy Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Membrane […]

For research use only. We do not sell to patients. Cyproheptadine CAS No. : 129-03-3 Biological Activity：Cyproheptadine is a potent and orally active 5-HT2A receptor antagonist, with antidepressant and antiserotonergic effects. Cyproheptadine has antiplatelet and thromboprotective activities. Cyproheptadine can be used for the research of thromboembolic disorders[2]. Research Area：Neurological Disease|Cardiovascular Disease Targets：5-HT Receptor|Apoptosis Related Small […]

For research use only. We do not sell to patients. ERα antagonist 1 CAS No. : 2762423-09-4 Biological Activity：ERα antagonist 1 (Compound 19d) is a potent, selective, covalent estrogen receptor α (ERα) antagonist. ERα antagonist 1 induces apoptosis and cell cycle G0/G1 phase arrest in MCF-7 cells. Research Area：Cancer Targets：Estrogen Receptor/ERR|Apoptosis Related Small Molecules:Physalin A;Bomedemstat […]

For research use only. We do not sell to patients. W146 TFA CAS No. : 909725-62-8 Biological Activity：W146 TFA is a selective antagonist of sphingosine-1-phosphate receptor 1 (S1PR1) with an EC50 value of 398 nM. Research Area：Cancer|Metabolic Disease Targets：LPL Receptor|Apoptosis Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor […]

For research use only. We do not sell to patients. Sertindole-d4 CAS No. : 1794737-42-0 Biological Activity：Sertindole-d4 (Lu 23-174-d4) is the deuterium labeled Sertindole. Sertindole, a neuroleptic, is one of the newer antipsychotic medications available[2]. Research Area：Neurological Disease|Cancer Targets：Dopamine Receptor|Adrenergic Receptor|5-HT Receptor|Autophagy Related Small Molecules:F 13714;Alizapride hydrochloride;Thioproperazine;Mosapride-d5;Todralazine;Bromopride-d3;ARC 239 dihydrochloride;Nuciferine;Yohimbine;Glaucine;Salbutamol;Renzapride;SB-277011 dihydrochloride;BI-167107;LY 344864 racemate;Harmine hydrochloride;Talibegron hydrochloride;MIF-1 TFA;Valerenic […]

For research use only. We do not sell to patients. Fimasartan-d6 Biological Activity：Fimasartan-d6 is deuterium labeled Fimasartan. Research Area：Cardiovascular Disease|Endocrinology Targets：Angiotensin Receptor|Apoptosis Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor 3;Xevinapant;Mangiferin;Cambinol;Antioxidant agent-5;Apoptosis inducer 9;Bafetinib;Cyclovirobuxine D;STAT3-IN-10;Rigosertib sodium Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  […]