Tag: Inducer|Agonist

For research use only. We do not sell to patients. N6-Benzyladenosine CAS No. : 4294-16-0 Biological Activity：N6-Benzyladenosine is an adenosine receptor agonist, has a cytoactive activity. N6-Benzyladenosine arrests cell cycle at G0/G1 phase and induces cell apoptosis. N6-Benzyladenosine also exerts inhibitory effect on T. gondii adenosine kinase and glioma–[5]. Research Area：Cancer|Inflammation/Immunology Targets：Adenosine Receptor|Apoptosis Related Screening […]

For research use only. We do not sell to patients. Bexarotene CAS No. : 153559-49-0 Biological Activity：Bexarotene (LGD1069) is a high-affinity and selective retinoid X receptors (RXR) agonist with EC50s of 33, 24, 25 nM for RXRα, RXRβ, and RXRγ, respectively. Bexarotene shows limited affinity for RAR receptors (EC50 >10000 nM)[2][3]. Bexarotene can be used for the research of cutaneous […]

For research use only. We do not sell to patients. PSB 0474 CAS No. : 917567-60-3 Biological Activity：PSB 0474 (3-phenacyl-UDP) is a selective and potent P2Y6 receptor agonist with an EC50 of 70 nM. PSB 0474 inhibits cell proliferation, increases NO release in astrocytes and microglia cells. PSB 0474 induces astrocytes apoptosis[2]. Research Area：Neurological Disease […]

For research use only. We do not sell to patients. BR102375 CAS No. : 2366255-59-4 Biological Activity：BR102375 is a non-TZD peroxisome proliferator-activated receptor γ (PPAR γ) full agonist for the treatment of type 2 diabetes, reveals EC50 value of 0.28 μM and Amax ratio of 98%. Research Area：Metabolic Disease Targets：PARP|Apoptosis Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase […]

For research use only. We do not sell to patients. Fenoldopam mesylate CAS No. : 67227-57-0 Biological Activity：Fenoldopam mesylate (SKF-82526) is a D1 receptor agonist and a novel lysine-specific demethylase 1 (LSD1) inhibitor (IC50=0.8974 μM). Fenoldopam mesylate shows anti-hypertensive effects, anti-cancer cell proliferation activity and can induce cells apoptosis[2][3]. Research Area：Cancer|Cardiovascular Disease Targets：Dopamine Receptor|Apoptosis Related […]

For research use only. We do not sell to patients. Norepinephrine bitartrate monohydrate CAS No. : 108341-18-0 Biological Activity：Norepinephrine (Levarterenol; L-Noradrenaline) bitartrate monohydrate is a potent adrenergic receptor (AR) agonist. Norepinephrine activates α1, α2, β1 receptors[2][3][4]. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor|Autophagy|Endogenous Metabolite Related Screening Libraries:Natural Product Library Plus;Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;Bioactive […]

For research use only. We do not sell to patients. Rilmenidine-d4 CAS No. : 85047-14-9 Biological Activity：Rilmenidine-d4 is the deuterium labeled Rilmenidine. Rilmenidine, an innovative antihypertensive agent, is an orally active, selective I1 imidazoline receptor agonist. Rilmenidine is an alpha 2-adrenoceptor agonist. Rilmenidine induces autophagy. Rilmenidine acts both centrally by reducing sympathetic overactivity and in […]

For research use only. We do not sell to patients. Octreotide CAS No. : 83150-76-9 Biological Activity：Octreotide (SMS 201-995) is a somatostatin receptor agonist and synthetic octapeptide endogenous somatostatin analogue. Octreotide (SMS 201-995) can bind to the somatostatin receptor and mainly subtypes 2, 3, and 5, increases Gi activity, and reduces intracellular cAMP production. Octreotide […]

For research use only. We do not sell to patients. Dienogest-d5 Biological Activity：Dienogest-d5 is deuterium labeled Dienogest. Research Area：Endocrinology|Cancer Targets：Autophagy|Progesterone Receptor|Apoptosis Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Gestonorone Capronate;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor 3;Xevinapant;Mangiferin;Cambinol;Antioxidant agent-5;Apoptosis inducer 9;Bafetinib;Cyclovirobuxine D;STAT3-IN-10 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  |  […]

For research use only. We do not sell to patients. Ankaflavin CAS No. : 50980-32-0 Biological Activity：Ankaflavin, isolated from Monascus-Fermented red rice, is an orally active PPARγ agonist. Ankaflavin exhibits selective cytotoxic effect and induces cell death through apoptosis on cancer cells. Ankaflavin has anti-inflammatory, anti-cancer, antiatherosclerotic, and hypolipidemic effects[2]. Research Area：Cancer|Inflammation/Immunology Targets：PPAR|Apoptosis Related Screening […]