Tag: Antagonist|Inhibitor|Modulator

For research use only. We do not sell to patients. Clozapine CAS No. : 5786-21-0 Biological Activity：Clozapine (HF 1854) is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors. Clozapine is a potent antagonist of dopamine D2 with a Ki of 75 nM. Clozapine inhibits the muscarinic […]

For research use only. We do not sell to patients. Clozapine-d8 CAS No. : 1185053-50-2 Biological Activity：Clozapine-d8 (HF 1854-d8) is the deuterium labeled Clozapine. Clozapine is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors[2][3][4]. Research Area：Neurological Disease Targets：Dopamine Receptor|Adrenergic Receptor|5-HT Receptor|mAChR Related Small Molecules:VU0357017 hydrochloride;F 13714;Alizapride […]

For research use only. We do not sell to patients. Aurintricarboxylic acid CAS No. : 4431-00-9 Biological Activity：Aurintricarboxylic acid is a nanomolar-potency, allosteric antagonist with selectivity towards αβ-methylene-ATP-sensitive P2X1Rs and P2X3Rs, with IC50s of 8.6 nM and 72.9 nM for rP2X1R and rP2X3R, respectively. Aurintricarboxylic acid is a potent anti-influenza agent by directly inhibiting the […]

For research use only. We do not sell to patients. Clozapine-d4 CAS No. : 204395-52-8 Biological Activity：Clozapine-d4 (HF 1854-d4) is the deuterium labeled Clozapine. Clozapine is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors[2][3][4][5]. Research Area：Neurological Disease Targets：Dopamine Receptor|Adrenergic Receptor|5-HT Receptor|mAChR Related Small Molecules:VU0357017 hydrochloride;F 13714;Alizapride […]