Tag: Antagonist

For research use only. We do not sell to patients. Methyllycaconitine citrate CAS No. : 351344-10-0 Biological Activity：Methyllycaconitine citrate is a specific antagonist of α7 neuronal nicotinic acetylcholine receptor (α7nAChR). Research Area：Neurological Disease Targets：nAChR Related Screening Libraries:Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor Compound Library;Anti-Parkinson’s Disease Compound Library;Neurodegenerative Disease-related Compound […]

For research use only. We do not sell to patients. BAY-6672 CAS No. : 2247517-53-7 Biological Activity：BAY-6672 is a potent and selective human Prostaglandin F (FP) receptor antagonist with an IC50 value of 11 nM. Research Area：Others Targets：Prostaglandin Receptor Related Small Molecules:Omidenepag isopropyl;DG-041;8-Isoprostaglandin E2;trans-Isoferulic acid;GSK-269984A;KMN-80;SC 51089;p-Hydroxycinnamic acid;Pexopiprant;Dinoprost;Sulprostone;Prostaglandin E2;CAY10471 Racemate;Fevipiprant;TG6-10-1;Cicaprost;ER-819762;MRE-269-d6;ONO-8130;KAG-308;KF 13218;Prostaglandin E2-d4 Trending products：Recombinant Proteins  |  […]

For research use only. We do not sell to patients. Diphenhydramine CAS No. : 58-73-1 Biological Activity：Diphenhydramine is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB)[2]. Research Area：Inflammation/Immunology|Cancer Targets：Histamine Receptor|Bacterial|Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide N-oxide;3-Hydroxyglutaric acid-d5;DPPC-d62;SDMA-d6;2-Mercaptobenzothiazole;Sandramycin;LLO (91-99);N-Acetyl-L-glutamic acid-d5;Gepotidacin;(3R,5S)-3-Hydroxy Cotinine-d3;Biliverdin hydrochloride;Oritavancin;Azlocillin sodium salt;D-Glucose-13C,d1-3;2,3-Diaminopropionic acid hydrochloride;Docosanoic […]

For research use only. We do not sell to patients. Mavoglurant racemate CAS No. : 1636881-61-2 Biological Activity：Mavoglurant racemate (AFQ-056 racemate) is the racemate of Mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Research Area：Neurological Disease Targets：mGluR Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:LY3020371 hydrochloride;ZJ43;FPTQ;(S)-MCPG;mGluR2 modulator 1;VU6010572;DFMTI;JNJ16259685;Auglurant;FITM;(-)-Camphoric acid;LY367385 hydrochloride;Cinnabarinic acid;LY379268;AZD 9272;mGluR2 antagonist […]

For research use only. We do not sell to patients. UNC4976 Biological Activity：UNC4976 is a positive allosteric modulator (PAM) peptidomimetic of CBX7 chromodomain binding to nucleic acids. UNC4976 simultaneously antagonizes H3K27me3-specific recruitment of CBX7 to target genes while increasing non-specific binding to DNA and RNA. Research Area：Cancer Targets：Histone Methyltransferase Related Small Molecules:EEDi-5285;EZH2-IN-2;BIX-01294;SGC707;(S)-HH2853;G9a-IN-1;MS1943;OTS186935 hydrochloride;MS8815;(R)-HH2853;EPZ020411;Furamidine dihydrochloride;EZH2-IN-12;UNC0642;MU1656;Chaetocin;UNC0646;UNC0224;MRK-740;SMYD2-IN-1;PRMT5-IN-21;Sinefungin;MM-401;SETDB1-TTD-IN-1;Dot1L-IN-2;PRMT5-IN-10;PRMT1-IN-1 Trending […]

For research use only. We do not sell to patients. Arotinolol CAS No. : 68377-92-4 Biological Activity：Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand 125I-ICYP to 5HT1B-serotonergic receptor sites[2]. Arotinolol is an antihypertensive agent for the treatment of a variety of […]

For research use only. We do not sell to patients. Sulpiride CAS No. : 15676-16-1 Biological Activity：Sulpiride is a D2 receptor a antagonist, an atypical antipsychotic drug of the benzamide class, used mainly in the treatment of psychosis associated with schizophrenia and major depressive disorder, and sometimes used in low dosage to treat anxiety and […]

For research use only. We do not sell to patients. Ondansetron-d3 hydrochloride CAS No. : 1346605-02-4 Biological Activity：Ondansetron-d3 (GR 38032-d3) hydrochloride) is the deuterium labeled Ondansetron hydrochloride. Ondansetron hydrochloride (GR 38032 hydrochloride) is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy[2]. Research Area：Neurological Disease Targets：5-HT Receptor […]

For research use only. We do not sell to patients. JNJ-47965567 CAS No. : 1428327-31-4 Biological Activity：JNJ-47965567 is a centrally permeable, high-affinity, selective P2X7 antagonist, with pKis of 7.9 and 8.7 for human and rat P2X7, respectively. JNJ-47965567 can be used to probe the role of central P2X7 in rodent models of CNS pathophysiology. Research […]

For research use only. We do not sell to patients. ABT-239 CAS No. : 460746-46-7 Biological Activity：ABT-239 is a novel, highly efficacious, non-imidazole class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist.  Research Area：Neurological Disease|Endocrinology Targets：TRP Channel|Histamine Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Membrane Transporter/Ion Channel […]