Tag: Agonist|Antagonist|Inhibitor

For research use only. We do not sell to patients. RG-12525 CAS No. : 120128-20-3 Biological Activity：RG-12525 is a a specific, competitive and orally effective antagonist of the peptidoleukotrienes, LTC4, LTD4 and LTE4, inhibiting LTC4-, LTD4- and LTE4-inducd guinea pig parenchymal strips contractions, with IC50s of 2.6 nM, 2.5 nM and 7 nM, respectively; RG-12525 […]

For research use only. We do not sell to patients. SCH-23390 maleate CAS No. : 87134-87-0 Biological Activity：SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively. SCH-23390 maleate is a potent and high efficacy human 5-HT2C […]