Tag: Agonist

For research use only. We do not sell to patients. Retinoic acid (GMP) CAS No. : 302-79-4 Biological Activity：Retinoic acid (Vitamin A acid) (GMP) is Retinoic acid (HY-14649) produced by using GMP guidelines. GMP small molecules works appropriately as an auxiliary reagent for cell therapy manufacture. Retinoic acid is an agonist of RAR nuclear receptors[2][3][4][5][6]. […]

For research use only. We do not sell to patients. Prucalopride-13C,d3 CAS No. : 2140306-00-7 Biological Activity：Prucalopride-13C,d3 is the 13C- and deuterium labeled Prucalopride. Research Area：Neurological Disease Targets：5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Nuciferine;Renzapride;LY 344864 racemate;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Tetrahydro-β-carboline;CP-809101;Volinanserin-d4 hydrochloride;Masupirdine free base;BRL-15572 dihydrochloride;LY393558;Brexpiprazole S-oxide Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  […]

For research use only. We do not sell to patients. SLIGRL-NH2 TFA Biological Activity：SLIGRL-NH2 TFA (Protease-Activated Receptor-2 Activating Peptide TFA) is an agonist of Protease-Activated Receptor-2 (PAR-2). Research Area：Inflammation/Immunology Targets：Protease Activated Receptor (PAR) Related Small Molecules:ENMD-1068 hydrochloride;Atopaxar hydrobromide;SCH79797 dihydrochloride;AC-55541;TRAP-6-IN-1;TRAP-6 amide TFA;I-191;ML354;Parstatin(human);UDM-001651;AZ8838;Protease-Activated Receptor-1, PAR-1 Agonist;TFLLR-NH2(TFA);tcY-NH2;VKGILS-NH2 TFA;2-Furoyl-LIGRLO-amide TFA;Protease-Activated Receptor-1 antagonist 1;GB-110;Protease-Activated Receptor-1 antagonist 2;RWJ-56110 dihydrochloride;Trypsin;TRAP-6;Protease-Activated Receptor-3 (PAR-3) (1-6), human […]

For research use only. We do not sell to patients. Remlarsen CAS No. : 1848266-71-6 Biological Activity：Remlarsen (MRG-201), a miR-29b mimic, acts a miR-29b agonist. Remlarsen has the potential for preventiong formation of a fibrotic scar or cutaneous fibrosis. Research Area：Inflammation/Immunology Targets：MicroRNA Related Small Molecules:(R)-Camptothecin-d5;Targaprimir-96 TFA;Lin28-let-7a antagonist 1;Camptothecin;Miravirsen;microRNA-21-IN-2;MIR96-IN-1;Gypenoside LI;Aurintricarboxylic acid;PIN1 inhibitor 2;LIN28 inhibitor LI71;Pseudoprotodioscin;Cl-amidine TFA;SID […]

For research use only. We do not sell to patients. Nalfurafine CAS No. : 152657-84-6 Biological Activity：Nalfurafine (TRK-820) is a potent selective and orally active G protein-biased kappa opioid receptor (KOR)-agonist with high translational potential. Nalfurafine (TRK-820) enhances the therapeutic potential of MOR-targeting analgesics, has the potential for uremic pruritis treatment[2]. Research Area：Neurological Disease Targets：Opioid […]

For research use only. We do not sell to patients. Siponimod hemifumarate CAS No. : 1234627-85-0 Biological Activity：Siponimod (BAF-312) hemifumarate is a potent and selective sphingosine-1-phosphate (S1P) receptor modulator. Siponimod hemifumarate is selective for S1P1 and S1P5 receptors over S1P2, S1P3, and S1P4 (EC50s of 0.39, 0.98, >10000, >1000, and 750 nM, respectively). Siponimod hemifumarate […]

For research use only. We do not sell to patients. NS 9283 CAS No. : 913830-15-6 Biological Activity：NS9283 is a positive positive allosteric modulator of (α4)3(β2)2 nicotinic ACh receptors. NS9283 can be used in a series of neurological conditions such as attention deficit hyperactivity disorder (ADHD), schizophrenia, Parkinson’s disease and Alzheimer’s disease. Research Area：Neurological Disease […]

For research use only. We do not sell to patients. CP-809101 CAS No. : 479683-64-2 Biological Activity：CP-809101 is a potent and highly selective 5-HT2C receptor agonist, with pEC50s of 9.96, 7.19 and 6.81 M for human 5HT2C, 5HT2B and 5HT2A receptor. CP-809101 inhibits conditioned avoidance responding in rats and antagonizes both PCP (phencyclidine hydrochloride)- and […]

For research use only. We do not sell to patients. Tizanidine-d4 hydrochloride CAS No. : 1188263-51-5 Biological Activity：Tizanidine-d4 (hydrochloride) is deuterium labeled Tizanidine (hydrochloride). Research Area：Cancer|Neurological Disease|Endocrinology Targets：Adrenergic Receptor Related Small Molecules:Todralazine;ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Talibegron hydrochloride;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR agonist 1;Tulobuterol;AGN 192836;KUC-7322;Oxyfedrine;Urapidil hydrochloride;Detomidine hydrochloride;Oxprenolol-d7 hydrochloride;Nicergoline;Synephrine hemitartrate;ADRA1D receptor antagonist 1;Solabegron Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  […]

For research use only. We do not sell to patients. L-803087 TFA CAS No. : 1786412-46-1 Biological Activity：L-803087 TFA is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM. L-803087 TFA is >280-fold more selective for sst4 receptor than other somatostatin receptors. L-803087 TFA facilitates AMPA-mediated hippocampal synaptic responses in […]