Tag: Agonist

For research use only. We do not sell to patients. Grifolic acid CAS No. : 80557-12-6 Biological Activity：Grifolic acid is a phenolic compound that is first extracted from the mushroom Albatrellus confluens. Grifolic acid acts as an agonist of the free fatty acid receptor (FFAR4/GPR120). Research Area：Inflammation/Immunology Targets：Free Fatty Acid Receptor Related Small Molecules:GW-1100;Ginsenoside Rb2;AP5;GPR40 […]

For research use only. We do not sell to patients. PPARγ agonist 7 CAS No. : 2569295-93-6 Biological Activity：PPARγ agonist 7 (Compound 3a) is a potent and selective agonist of PPARγ. PPARγ agonist 7 promotes adiponectin production in human bone marrow mesenchymal stem cells (hBM-MSCs) as a novel PPARγ full agonist (EC50, 4.34 μM). Research […]

For research use only. We do not sell to patients. (Rac)-Razpipadon CAS No. : 1643462-93-4 Biological Activity：PW0464, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP). Research Area：Neurological Disease Targets：Dopamine Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor […]

For research use only. We do not sell to patients. Budesonide-d8 CAS No. : 1105542-94-6 Biological Activity：Budesonide-d8 is the deuterium labeled Budesonide. Budesonide, an inhaled glucocortical steroid, is an orally active glucocorticoid receptor agonist. Budesonide decreases the size of lung tumors, reverses DNA hypomethylation and modulates mRNA expression of genes. Budesonide is an anti-inflammatory agent […]

For research use only. We do not sell to patients. MIPS521 CAS No. : 1146188-19-3 Biological Activity：MIPS521 is a positive allosteric modulator of adenosine A1 receptor (A1AR). MIPS521 also has a lower A1R allosteric affinity (pKB=4.95; KB=11 μM). MIPS521 exhibits pain-relieving effects in vivo through modulation of the increased levels of endogenous adenosine[2]. Research Area：Neurological Disease […]

For research use only. We do not sell to patients. Budesonide impurity C CAS No. : 1040085-99-1 Biological Activity：Budesonide impurity C is an impurity of Budesonide. Budesonide, an inhaled glucocortical steroid, is an orally active glucocorticoid receptor agonist[2]. Research Area：Cancer|Inflammation/Immunology Targets：Glucocorticoid Receptor Related Small Molecules:Deflazacort-D5;Glucocorticoid receptor agonist-2;AZD2906;Beclometasone dipropionate;ORIC-101;Clobetasone butyrate;Cortisone-d2;Clobetasone butyrate-d7;Cortisone-13C3;Glucocorticoid receptor agonist;Cortodoxone-d2;Hydrocortisone aceponate;Glucocorticoid receptor-IN-2;OP-3633;GW-870086;Nenocorilant;Hydrocortisone cypionate;Corticosterone-d8;21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione;Deflazacort-d5-1;Mapracorat;Hydrocortisone-d4;Hydrocortisone […]

For research use only. We do not sell to patients. S1p receptor agonist 2 CAS No. : 1354908-17-0 Biological Activity：S1p receptor agonist 2 (compound 1) is an agonist of S1P5 receptor, exhibits selectivity over the S1P1 and/or S1P3 receptors. S1p receptor agonist 2 can be used for endogenous SIP signaling system research, and alleviating or […]

For research use only. We do not sell to patients. Prednisolone CAS No. : 50-24-8 Biological Activity：Prednisolone is a potent, orally active corticosteroid and a glucocorticoid. Prednisolone possesses about four times the anti-inflammatory activity of hydrocortisone while causing less salt and water retention. Prednisolone can be used for ocular, anti-inflammatory research[2]. Research Area：Endocrinology|Inflammation/Immunology Targets：Glucocorticoid Receptor|Endogenous […]

For research use only. We do not sell to patients. KMN-80 CAS No. : 1628759-75-0 Biological Activity：KMN-80, a derivative of PGE1 (HY-B0131), is a selective and potent agonist of EP4 receptor with an IC50 and a Ki of 3 nM and 2.35 nM, respectively. KMN-80 is against EP3 receptor with an IC50 of 1.4 μM […]

For research use only. We do not sell to patients. Velmupressin acetate CAS No. : 1647120-04-4 Biological Activity：Velmupressin (c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2) acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively. Research Area：Metabolic Disease Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl […]