Tag: Agonist

For research use only. We do not sell to patients. 1-Aminocyclobutanecarboxylic acid CAS No. : 22264-50-2 Biological Activity：1-Aminocyclobutanecarboxylic acid is a NMDA receptor partial agonist acting at the glycine site, NR1. Research Area：Neurological Disease Targets：iGluR Related Screening Libraries:Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor Compound Library;Protein-protein Interaction Inhibitor Library; Related […]

For research use only. We do not sell to patients. TLR8 agonist 5 CAS No. : 2413016-41-6 Biological Activity：TLR8 agonist 5 is a potent TLR8 agonist with an EC50 value of 20 nM for HEK-Blue hTLR8. TLR8 agonist 5 activates the immune response. Research Area：Inflammation/Immunology Targets：Toll-like Receptor (TLR) Related Small Molecules:C29;TMX-201;RS 09;ODN 20844;TLR7/8-IN-1;Sulfo-ara-F-NMN;TLR7/8 antagonist 1;Gardiquimod;PF-4878691;Tri(TLR4-IN-C34-PEG2-amide-PEG1)-amide-C3-COOH;Pepinh-TRIF […]

For research use only. We do not sell to patients. Triamcinolone acetonide-d7-1 Biological Activity：Triamcinolone acetonide-d7-1 is deuterium labeled Triamcinolone acetonide. Research Area：Inflammation/Immunology|Endocrinology|Cancer Targets：Glucocorticoid Receptor Related Small Molecules:Deflazacort-D5;Glucocorticoid receptor agonist-2;AZD2906;Beclometasone dipropionate;ORIC-101;Clobetasone butyrate;Cortisone-d2;Clobetasone butyrate-d7;Cortisone-13C3;Glucocorticoid receptor agonist;Cortodoxone-d2;Hydrocortisone aceponate;Glucocorticoid receptor-IN-2;OP-3633;GW-870086;Nenocorilant;Hydrocortisone cypionate;Corticosterone-d8;21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione;Deflazacort-d5-1;Mapracorat;Hydrocortisone-d4;Hydrocortisone acetate Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled […]

For research use only. We do not sell to patients. Uridine 5′-diphosphoglucose disodium salt CAS No. : 28053-08-9 Biological Activity：Uridine 5′-diphosphoglucose disodium salt (UDP-D-Glucose disodium salt) is the precursor of glucose-containing oligosaccharides, polysaccharides, glycoproteins, and glycolipids in animal tissues and in some microorganisms. Uridine-5′-diphosphoglucose is an agonist of the P2Y14 receptor, a neuroimmune system GPCR. […]

For research use only. We do not sell to patients. Talibegron hydrochloride CAS No. : 178600-17-4 Biological Activity：Talibegron hydrochloride (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect. Research Area：Cardiovascular Disease Targets：Adrenergic Receptor Related Small Molecules:Todralazine;ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR […]

For research use only. We do not sell to patients. APNEA CAS No. : 89705-21-5 Biological Activity：APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. Research Area：Neurological Disease Targets：Adenosine Receptor Related Screening Libraries:Natural Product-like Compound Library;Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Clinical Compound Library;Small Molecule Immuno-Oncology Compound […]

For research use only. We do not sell to patients. FG8119 CAS No. : 106447-61-4 Biological Activity：FG8119 is a novel benzodiazepine agonist extracted from patent US 4745112 A. Research Area：Neurological Disease Targets：GABA Receptor Related Small Molecules:SKF89976A hydrochloride;mGAT-IN-1;Alpidem;Valerenic acid;Picrotoxinin;Miltirone;Etifoxine-13C,d3;Adipiplon;Gabazine;Broflanilide;Fluxametamide;ONO-8590580;γ-Aminobutyric acid-d6;Ginsenoside Rc;Fipronil;p-Hydroxybenzaldehyde-13C;Lesogaberan hydrochloride;FG 7142;Isoguvacine hydrochloride;Guvacine ethyl ester;MRK-623;Rilmazafone;(-)-α-Pinene;Alpidem-d14;17-PA Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  […]

For research use only. We do not sell to patients. Chlormadinone acetate-d6-1 Biological Activity：Chlormadinone acetate-d6-1 is deuterium labeled Chlormadinone acetate. Research Area：Endocrinology Targets：Progesterone Receptor Related Small Molecules:Gestonorone Capronate;17α-Hydroxyprogesterone;Nestoron;Melengestrol acetate-d2;Asoprisnil-d3;Norgestrel-d6;Progesterone-13C2;Melengestrol acetate;Progesterone;Progesterone-13C5;PF-02413873;Chlormadinone acetate;Chlormadinone acetate-d6;ARD-61;Altrenogest Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  |  Oligonucleotides About Us: MedChemExpress […]

For research use only. We do not sell to patients. GLP-1R agonist 4 CAS No. : 2401894-26-4 Biological Activity：GLP-1R agonist 4 is a potent agonist of GLP-1R. Glucagon-like peptide-1 (GLP-1) is an intestinal hypoglycemic hormone secreted by L-cells in the lower gastrointestinal tract. GLP-1R agonist 4 has the potential for the research of diabetes (extracted […]

For research use only. We do not sell to patients. Denopamine CAS No. : 71771-90-9 Biological Activity：Denopamine ((R)-(-)-Denopamine) is an orally active, selective β1-adrenergic agonist. Denopamine prolongs survival in a murine model of congestive heart failure induced by viral myocarditis: suppression of tumor necrosis factor-α production in the heart. Cardiovascular effects. Research Area：Cardiovascular Disease Targets：Adrenergic […]