Tag: Agonist

For research use only. We do not sell to patients. RVD-Hpα TFA Biological Activity：RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM). […]

For research use only. We do not sell to patients. Salbutamol CAS No. : 18559-94-9 Biological Activity：Salbutamol is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease (COPD). Research Area：Neurological Disease|Endocrinology Targets：Adrenergic Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved […]

For research use only. We do not sell to patients. Renzapride CAS No. : 112727-80-7 Biological Activity：Renzapride (BRL 24924), a substituted benzamide, is a full 5-HT4 receptor agonist with a Ki value of 115 nM. Renzapride (BRL 24924) is also a 5HT2b and 5HT3 receptor antagonist. Renzapride could be used for constipation predominant irritable bowel […]

For research use only. We do not sell to patients. AC-262536 CAS No. : 870888-46-3 Biological Activity：AC-262536 is a selective and non-steroidal androgen receptor modulators (SARMs) with beneficial anabolic effects. AC-262536 exhibits potent agonist activity at the androgen receptor, with an affinity in the low nanomolar range (1-10 nM). Research Area：Metabolic Disease Targets：Androgen Receptor Related […]

For research use only. We do not sell to patients. β-Caryophyllene CAS No. : 87-44-5 Biological Activity：β-Caryophyllene is a CB2 receptor agonist. Research Area：Cancer|Infection|Neurological Disease Targets：Endogenous Metabolite|Cannabinoid Receptor Related Screening Libraries:Natural Product Library Plus;Bioactive Compound Library Plus;Anti-Infection Compound Library;GPCR/G Protein Compound Library;Metabolism/Protease Compound Library;Neuronal Signaling Compound Library;Natural Product Library;Anti-Cancer Compound Library;Human Endogenous Metabolite Compound Library;Lipid […]

For research use only. We do not sell to patients. Cinacalcet-d3 hydrochloride Biological Activity：Cinacalcet-D3 (AMG 073-D3) hydrochloride is the deuterium labeled Cinacalcet (hydrochloride). Cinacalcet hydrochloride (AMG-073 hydrochloride) is an orally active, allosteric agonist of Ca receptor (CaR), used for cardiovascular disease treatment. Research Area：Cardiovascular Disease Targets：CaSR|Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide N-oxide;3-Hydroxyglutaric acid-d5;DPPC-d62;SDMA-d6;2-Mercaptobenzothiazole;N-Acetyl-L-glutamic acid-d5;(3R,5S)-3-Hydroxy […]

For research use only. We do not sell to patients. BI-167107 CAS No. : 1202235-68-4 Biological Activity：BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. Research Area：Cancer|Neurological Disease|Endocrinology Targets：Adrenergic Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound […]

For research use only. We do not sell to patients. LY 344864 racemate CAS No. : 186543-64-6 Biological Activity：LY 344864 racemate is a 5-HT1F receptor agonist extracted from patent US 5708187 A. Research Area：Neurological Disease Targets：5-HT Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor Compound Library;Anti-Alzheimer’s Disease Compound Library;Anti-Obesity […]

For research use only. We do not sell to patients. Retinoic acid CAS No. : 302-79-4 Biological Activity：Retinoic acid is a metabolite of vitamin A that plays important roles in cell growth, differentiation, and organogenesis. Retinoic acid is a natural agonist of RAR nuclear receptors, with IC50s of 14 nM for RARα/β/γ. Retinoic acid bind […]

For research use only. We do not sell to patients. Pancreatic Polypeptide, human CAS No. : 75976-10-2 Biological Activity：Pancreatic Polypeptide, human is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist. Research Area：Metabolic Disease|Endocrinology Targets：Neuropeptide Y Receptor Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:[D-Trp34]-Neuropeptide […]