Apabetalone

For research use only. We do not sell to patients.

Apabetalone

CAS No. : 1044870-39-4

Biological Activity:Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. The IC50s are 87 μM and 0.51 μM for BD1 and BD2, respectively.

Research Area:Cancer

Targets:Epigenetic Reader Domain|HIV

Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Anti-Infection Compound Library;Epigenetics Compound Library;Histone Modification Research Compound Library;Anti-Cancer Compound Library;Clinical Compound Library;Antiviral Compound Library;Drug Repurposing Compound Library;Reprogramming Compound Library;Anti-diabetic Compound Library;Anti-Blood Cancer Compound Library;Rare Diseases Drug Library;Protein-protein Interaction Inhibitor Library;Human Metabolite Library;

Related Small Molecules:RVX-297;BRD4 Inhibitor-19;HIV-1 TAT (48-60);Seletracetam lithium;HIV-IN-2;UNC6349 (Ket2);Curcumin;Triptonine B;GSK6853;GSK4028;FC131;Peritassine A;SR-0813;Flavopiridol;Inobrodib;TAT (48-57);FGI-106 tetrahydrochloride;(Z)-9-Propenyladenine;OF-1;I-CBP112;Decanoyl-RVKR-CMK TFA;ONX-0914 TFA

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