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Taletrectinib
CAS No. : 1505515-69-4
Biological Activity：Taletrectinib (DS-6051b) is a potent, orally active, and next-generation selective ROS1/NTRK inhibitor. Taletrectinib potently inhibits recombinant ROS1, NTRK1, NTRK2, and NTRK3 with IC50s of 0.207, 0.622, 2.28, and 0.98 nM, respectively. Taletrectinib also inhibits ROS1 G2032R and other Crizotinib-resistant ROS1 mutants[2].
Research Area：Cancer
Targets：ROS Kinase
Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Kinase Inhibitor Library;Protein Tyrosine Kinase Compound Library;Anti-Cancer Compound Library;Clinical Compound Library;Drug Repurposing Compound Library;Orally Active Compound Library;Anti-Lung Cancer Compound Library;Targeted Diversity Library;
Related Small Molecules:GGTI-2154 hydrochloride;MitoPQ;Entrectinib;WY-135;Anticancer agent 59;Uniconazole;Anticancer agent 76;Salvigenin;ROS kinases-IN-1;Anticancer agent 58;AChE/BChE/BACE-1-IN-2;Merestinib;Repotrectinib;Lorlatinib;AChE/GSK-3β-IN-1;Keap1-Nrf2-IN-11;Phyltetralin;ROS kinases-IN-2;GGTI-2418;Capsanthin;F-1;Apogossypolone;Lorlatinib-13C,d3;AChE/BChE-IN-9
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