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Tetrabenazine Racemate

CAS No. : 718635-93-9

Biological Activity：Tetrabenazine Racemate (Ro 1-9569 Racemate) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).
(1) The reference for administration is 0.25-0.75 mg/kg IP
(2) Injections of tetrabenazine into accumbens core also reduced FR5 lever pressing and increased chow intake.
(3) Tetrabenazine (Racemate) reduced extracellular DA and altered DARPP-32 signaling in both substance-P- and enkephalin-containing accumbens neurons.
(4) Tetrabenazine (Racemate) inhibits locomotor activity and produces hypothermia upon systemic administration in rats and mice.

Research Area：Neurological Disease

Targets：Monoamine Transporter

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