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Dersimelagon

CAS No. : 1835256-48-8

Biological Activity：Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC₅₀ values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon shows good affinity for hMC1R and hMC4R with K_i values of 2.26, 32.9 nM, respectively. Dersimelagon can be used for the research of skin pigmentation^{[1]^{^{[2]^.}}}

Research Area：Metabolic Disease

Targets：Melanocortin Receptor

Related Small Molecules:Bremelanotide;MSG606 TFA;Resomelagon;Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA;Terrein;γ1-MSH TFA;SNT-207707;PF-07258669;THIQ;ACTH (11-24) (acetate);JKC363 TFA;PG-931 TFA;[D-Trp8]-γ-MSH;MC-4R Agonist 1;ACTH (1-17);SNT-207858 free base;Lys-γ3-MSH(human);Nonapeptide-1;HS024 TFA;Adrenocorticotropic Hormone (ACTH) (4-10), human;SHU 9119;Adrenocorticotropic Hormone (ACTH) (1-39), human(TFA);(p-Iodo-Phe7)-ACTH (4-10)

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