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PD176252
CAS No. : 204067-01-6
Biological Activity：PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.
Research Area：Cancer
Targets：Bombesin Receptor
Related Screening Libraries:Covalent Screening Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Cancer Compound Library;Covalent Screening Library;
Related Small Molecules:Bombesin;RC-3095;BA 1;BIM-26226;ML-18;Kuwanon H;MK-5046;Litorin;Ranatensin;Kuwanon G;PD 168368
Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
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