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Relugolix

CAS No. : 737789-87-6

Biological Activity：Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC₅₀=0.33 nM) and monkey receptor (IC₅₀=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al^[2].

Research Area：Cancer|Endocrinology

Targets：GnRH Receptor

Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;FDA-Approved Drug Library;Anti-Cancer Compound Library;Drug Repurposing Compound Library;Endocrinology Compound Library;Anti-COVID-19 Compound Library;Orally Active Compound Library;FDA Approved & Pharmacopeial Drug Library;FDA-Approved Anticancer Drug Library;Human Metabolite Library;Anti-Prostate Cancer Compound Library;

Related Small Molecules:(R)-Elagolix;Linzagolix;Relugolix-d6;[D-Ala6]-LH-RH;Teverelix;Alarelin Acetate;[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide;Kisspeptin 13;opigolix;sGnRH-A;Lecirelin;GnRH-R antagonist 1;Ozarelix;LH-RH (7-10);BAY-298;Acyline;GnRH-I;Lamprey LH-RH I;BAY-784;BAY 1214784;GnRH antagonist 2;[D-Lys6]-LH-RH

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