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Pimethixene maleate
CAS No. : 13187-06-9
Biological Activity：Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent.
Pimethixene maleate is a highly potent antagonist of 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors, with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively.
Research Area：Neurological Disease|Endocrinology
Targets：5-HT Receptor|Histamine Receptor
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Related Small Molecules:F 13714;Mosapride-d5;Nuciferine;Tripelennamine;Renzapride;Brompheniramine-d6 maleate;LY 344864 racemate;Samelisant;Harmine hydrochloride;Chlorphenoxamine;Valerenic acid;H3 receptor-MO-1;Diphenhydramine;Arotinolol;ABT-239;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride
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