H4R antagonist 1

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H4R antagonist 1

CAS No. : 1429375-54-1

Biological Activity:H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R.

Research Area:Inflammation/Immunology|Endocrinology

Targets:Histamine Receptor

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