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ELN-441958

CAS No. : 913064-47-8

Biological Activity：ELN-441958 is a potent, neutral, competitive and selective bradykinin B₁ receptor antagonist with a K_i of 0.26 nM against native human bradykinin B₁ receptor. ELN-441958 has high oral bioavailability, and has low CNS exposure in the mouse.

Research Area：Endocrinology|Inflammation/Immunology

Targets：Bradykinin Receptor

Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Endocrinology Compound Library;Neurotransmitter Receptor Compound Library;Targeted Diversity Library;

Related Small Molecules:Icatibant acetate;Retrobradykinin;Bombinakinin M;[Tyr8] Bradykinin;Bradykinin (2-9);Deucrictibant;Fasitibant chloride;WIN 64338 hydrochloride;Bradykinin (1-7);Lys-[Hyp3]-Bradykinin;Bradykinin (1-6);[Hyp3]-Bradykinin;[Des-Arg9]-Bradykinin acetate;Lys-[Des-Arg9]Bradykinin TFA;Lobradimil;Bradykinin;Bradykinin (1-5);FR167344 free base;SSR240612;Fulimetibant;B 9430;Bradykinin (1-3)

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