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GSK256073
CAS No. : 862892-90-8
Biological Activity：GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia[2]. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
Research Area：Metabolic Disease
Targets：GPR109A
Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Clinical Compound Library;Drug Repurposing Compound Library;Anti-diabetic Compound Library;Targeted Diversity Library;
Related Small Molecules:MK-0354;MK-6892;GPR109 receptor agonist-1;Acifran
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