RG108

For research use only. We do not sell to patients.

RG108

CAS No. : 48208-26-0

Biological Activity:RG108 (N-Phthalyl-L-tryptophan) is a non-nucleoside DNA methyltransferases (DNMTs) inhibitor (IC50=115 nM) that blocks the DNMTs active site. RG108 (N-Phthalyl-L-tryptophan) causes demethylation and reactivation of tumor suppressor genes, but it does not affect the methylation of centromeric satellite sequences[2][3].

Research Area:Cancer

Targets:DNA Methyltransferase

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