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Tolvaptan

CAS No. : 150683-30-0

Biological Activity：Tolvaptan is a selective, competitive and orally active vasopressin receptor 2 (V₂R) antagonist with an IC₅₀ of 1.28 μM for the inhibition of arginine vasopressin (AVP)-induced platelet aggregation. Tolvaptan induces cell apoposis and affects cell cycle. Tolvaptan can be used for the research of hyponatremia^[2].

Research Area：Cardiovascular Disease|Endocrinology|Cancer

Targets：Autophagy|Vasopressin Receptor

Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;FDA-Approved Drug Library;Anti-Cancer Compound Library;Autophagy Compound Library;Drug Repurposing Compound Library;Anti-Cardiovascular Disease Compound Library;Endocrinology Compound Library;Anti-COVID-19 Compound Library;NMPA-Approved Drug Library;Orally Active Compound Library;FDA Approved & Pharmacopeial Drug Library;Drug-Induced Liver Injury (DILI) Compound Library;Targeted Diversity Library;Rare Diseases Drug Library;Children’s Drug Library;EMA-Approved Drug Library;FDA-Approved Anticancer Drug Library;Coagulation and Anti-coagulation Compound Library;

Related Small Molecules:Lixivaptan;Mozavaptan hydrochloride;Balovaptan;Big Endothelin-1 (1-38), human;WAY-151932;Felypressin;Antagonist G TFA;Mozavaptan-d6;SKF 100398;Fedovapagon;L-371,257;Argipressin;D[LEU4,LYS8]-VP;d[Cha4]-AVP;RG7713;TASP0390325;Terlipressin-d5;SRX246;Terlipressin acetate;SR 49059;Big Endothelin-1 (1-39), porcine

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