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RLX-33
CAS No. : 2784577-71-3
Biological Activity：RLX-33 is a potent, selective and blood-brain barrier (BBB) penetrant relaxin family peptide 3 (RXFP3) antagonist, also blocks relaxin-3-induced ERK1/2 phosphorylation, with IC50 values of 2.36 μM for RXFP3, 7.82 and 13.86 μM for ERK1 and ERK2 phosphorylation, respectively. RLX-33 can block the stimulation of food intake induced by the RXFP3-selective agonist R3/I5 in rats. RLX-33 can be used for the research of metabolic syndrome.
Research Area：Metabolic Disease
Targets：ERK
Related Screening Libraries:Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Kinase Inhibitor Library;MAPK Compound Library;Stem Cell Signaling Compound Library;CNS-Penetrant Compound Library;Anti-Aging Compound Library;Oxygen Sensing Compound Library;Glutamine Metabolism Compound Library;Angiogenesis-Related Compound Library;
Related Small Molecules:Corynoxeine;Temuterkib;CKLF1-C27;LM22B-10;ERK5-IN-4;Pachymic acid;MAP855;6-OAU;VX-11e;Pluripotin;2,5-Dihydroxyacetophenone;Astragaloside IV;ERK1/2 inhibitor 1;Longdaysin;[Tyr8] Bradykinin;Gypenoside L;ERK-IN-2;Omtriptolide;Chemerin-9 (149-157);MAPK-IN-1;SHR2415;Anti-inflammatory agent 31;PACAP-38 (31-38), human, mouse, rat TFA;AKT-IN-11;N-Salicyloyltryptamine;JWG-071
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