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Telcagepant

CAS No. : 781649-09-0

Biological Activity：Telcagepant (MK-0974) is an orally active calcitonin gene-related peptide (CGRP) receptor antagonist with K_is of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively.

Research Area：Neurological Disease

Targets：CGRP Receptor

Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Clinical Compound Library;Drug Repurposing Compound Library;Anti-COVID-19 Compound Library;Orally Active Compound Library;

Related Small Molecules:Vazegepant hydrochloride;Adrenomedullin (16-31), human;MK-3207 Hydrochloride;α-CGRP, rat;Cagrilintide acetate;HTL22562;SUN B8155;Adrenomedullin (11-50), rat;Rat CGRP-(8-37);Atogepant;β-CGRP, human TFA;Calcitonin (salmon);Calcitonin (human);α-CGRP(human);Galcanezumab;Olcegepant;Rimegepant;Calcitonin Gene Related Peptide (CGRP) II, rat;Ubrogepant;PHM-27 (human);Adrenomedullin (1-50), rat;CGRP antagonist 1;HCGRP-(8-37)

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