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Sigma-1 receptor antagonist 3
CAS No. : 1639220-17-9
Biological Activity：Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain.
Research Area：Neurological Disease
Targets：Sigma Receptor|Potassium Channel
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