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SSR240612
CAS No. : 464930-42-5
Biological Activity：SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist, with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.
Research Area：Metabolic Disease|Inflammation/Immunology|Endocrinology
Targets：Bradykinin Receptor
Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Endocrinology Compound Library;Orally Active Compound Library;Neurotransmitter Receptor Compound Library;
Related Small Molecules:Icatibant acetate;Retrobradykinin;Bombinakinin M;[Tyr8] Bradykinin;Bradykinin (2-9);Deucrictibant;Fasitibant chloride;WIN 64338 hydrochloride;ELN-441958;Bradykinin (1-7);Lys-[Hyp3]-Bradykinin;Bradykinin (1-6);[Hyp3]-Bradykinin;[Des-Arg9]-Bradykinin acetate;Lys-[Des-Arg9]Bradykinin TFA;Lobradimil;Bradykinin;Bradykinin (1-5);FR167344 free base;Fulimetibant;B 9430;Bradykinin (1-3)
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