Tasimelteon

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Tasimelteon

CAS No. : 609799-22-6

Biological Activity:Tasimelteon (BMS-214778) is an orally active and selective dual melatonin receptor agonist (DMRA). Tasimelteon has 2.1-4.4 times greater affinity for the MT2 receptor than for the MT1 receptor. Tasimelteon is a circadian regulator and has the potential for Non-24-Hour Sleep-Wake Disorder (Non-24)[2].

Research Area:Neurological Disease|Endocrinology

Targets:Melatonin Receptor

Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;FDA-Approved Drug Library;Drug Repurposing Compound Library;Endocrinology Compound Library;Anti-COVID-19 Compound Library;Orally Active Compound Library;FDA Approved & Pharmacopeial Drug Library;Drug-Induced Liver Injury (DILI) Compound Library;Rare Diseases Drug Library;EMA-Approved Drug Library;

Related Small Molecules:Melatonin-d3;Antidepressant agent 3;6-Chloromelatonin;DH97;TIK-301;N-Acetyltryptamine;Luzindole;ACH-000143;Antidepressant agent 4;Agomelatin-d3;UCM 608;4-P-PDOT;Piromelatine;8-M-PDOT;S26131;Melatonin-d7;2-Iodomelatonin

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