For research use only. We do not sell to patients.
Zeteletinib hemiadipate
CAS No. : 2375837-06-0
Biological Activity：Zeteletinib (BOS-172738; DS-5010) hemiadipate is an orally active, selective RET kinase inhibitor with nanomolar potency against RET and >300-fold selectivity against VEGFR2. Zeteletinib hemiadipate shows exquisite potency for the wild type RET, RETV804M/L gatekeeper mutants, and the most common oncogenic RET mutation M918T. Zeteletinib hemiadipate has potent antitumor activity[2][3].
Research Area：Cancer
Targets：RET|PDGFR
Related Small Molecules:Henatinib;Flumatinib mesylate;IHMT-TRK-284;RET-IN-18;PDGFRα/FLT3-ITD-IN-2;PP58;Chiauranib;Zeteletinib;ENMD-2076 Tartrate;AZD2932;RET-IN-5;AC710 Mesylate;Tyrosine kinase-IN-1;GSK3179106;Tandutinib;JNJ-10198409;SU4984;Pyrazoloadenine;SU4312;Avapritinib;MELK-8a;trans-Pralsetinib;PF 477736
Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
About Us:
- MedChemExpress (MCE) offers a wide range of high-quality research chemicals and biochemicals (novel life-science reagents, reference compounds and natural compounds) for scientific use；
- Structurally and synthetically diverse biologically active compounds；
- roduct quality is the key to our success and we take pride in offering only the highest-grade products.；
- We provide HNMR, LC-MS, HPLC, stability testing and activity assays of our products to clients.；
- Product identity, quality, purity and activity are assured by our robust quality control programs and procedures.；
- Customized order volume ranging from milligrams to kilograms scale；
Structurally and synthetically diverse biologically active compounds；
We provide customer-oriented services. To explore more, please contact us at [email protected]. Our team will gladly assist you.
