2023 - epigenetics modulation frontier

Antitrypanosomal agent 2

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Antitrypanosomal agent 2 CAS No. : 475626-30-3 Biological Activity：Antitrypanosomal agent 2 is a potent and selective trypanosoma brucei inhibitor. Research Area：Infection Targets：Parasite Related Small Molecules:(+)-Isopulegol;SR9186;Antileishmanial agent-2;Azlocillin sodium salt;SQ109;Trypanothione synthetase-IN-3;Pyrantel;α-Terpinene;Dehydrocorydaline;Niclosamide monohydrate;Febrifugine dihydrochloride;Antimalarial agent 15;Cycloguanil hydrochloride;Anti-infective agent 6;Morantel tartrate;Sulfiram;UCB7362;Retro-2;PfDHODH-IN-2;ML251 Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products […]

FLAG peptide

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. FLAG peptide CAS No. : 98849-88-8 Biological Activity：FLAG peptide is an eight amino acids peptide (Asp-Tyr-Lys-Asp-Asp-Asp-Asp-Lys) with an enterokinase-cleavage site; designed for antibody-mediated identification and purification of recombinant proteins. Research Area：Inflammation/Immunology Targets：Others Related Screening Libraries:Bioactive Compound Library Plus;Peptidomimetic Library; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole […]

GK563

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. GK563 CAS No. : 2351820-19-2 Biological Activity：GK563 is a selective Ca2+-independent phospholipase A2 (GVIA iPLA2) inhibitor with an IC50 value of 1 nM. GK563 is 22000 times more active against GVIA iPLA2 than GIVA cPLA2. GK563 reduces β-cell apoptosis induced by proinflammatory cytokines, raising the […]

Cinaciguat hydrochloride

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Cinaciguat hydrochloride CAS No. : 646995-35-9 Biological Activity：Cinaciguat hydrochloride is a potent soluble guanylate cyclase (GC) activator with EC50 of 15 nM in platelets. Research Area：Cardiovascular Disease Targets：Guanylate Cyclase Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Clinical […]

ZIKV-IN-4

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. ZIKV-IN-4 Biological Activity：ZIKV-IN-4 (compound 5b) is a low-cytotoxicity and acid-stable anti-ZIKV agent (EC50=3.49 μM). ZIKV-IN-4 effectively inhibits the activity of ZIKV NS5 MTase. Research Area：Infection Targets：Virus Protease Related Small Molecules:SRPIN340;Aminothiazole;CYP2C9/CYP2C19-IN-1;L-Lysine;L-Lysine-13C6,15N2,d9 dihydrochloride;4E2RCat;ESI-09;Tubacin;Lycorine;PCL 016;NGI-1;(-)-α-Pinene;Encephalitic alphavirus-IN-1;HCVcc-IN-1;L-Lysine-d4 hydrochloride;ZINC03129319;SARS-CoV-2 Mpro-IN-4;Palmatine;Ensitrelvir;NS2B/NS3-IN-6;NS2B/NS3-IN-4;L-Lysine-d9 hydrochloride;Hinokitiol;L-Lysine-15N-1 dihydrochloride Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]

(β-Ala8)-Neurokinin A (4-10)

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. (β-Ala8)-Neurokinin A (4-10) CAS No. : 127633-71-0 Biological Activity：(β-Ala8)-Neurokinin A (4-10), a neuropeptide, is a potent and selective NK-2 tachykinin receptor (Neurokinin Receptor) agonist. Research Area：Neurological Disease Targets：Neurokinin Receptor Related Small Molecules:Talnetant hydrochloride;Pavinetant;MEN11467;(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P;Vapreotide acetate;Rolapitant;Eprazinone dihydrochloride;Orvepitant maleate;Netupitant metabolite Monohydroxy Netupitant;SB-222200;Senktide;GR 87389;Hemokinin 1, human;Neurokinin A TFA;Imnopitant […]

Stauprimide

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Stauprimide CAS No. : 154589-96-5 Biological Activity：Stauprimide is a staurosporine analog that promotes embryonic stem cell (ESC) differentiation. Stauprimide is a non-broad spectrum inhibitor that binds to the MYC transcription factor NME2 and blocks its nuclear localization in ESCs, which results in down-regulation of MYC […]

5-Fluorouracil-d1

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. 5-Fluorouracil-d1 CAS No. : 90344-84-6 Biological Activity：5-Fluorouracil-d1 (5-FU-d1) is the deuterium labeled 5-Fluorouracil. 5-Fluorouracil (5-FU) is an analogue of uracil and a potent antitumor agent. 5-Fluorouracil affects pyrimidine synthesis by inhibiting thymidylate synthetase thus depleting intracellular dTTP pools. 5-Fluorouracil induces apoptosis and can be used […]

Neocurdione

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Neocurdione CAS No. : 108944-67-8 Biological Activity：Neocurdione is a hepatoprotective sesquiterpene isolated from Curcuma zedoaria rhizome. Neocurdione exerts potent effect on D-galactosamine- (D-Gain) and lipopolysaccharide- (LPS) induced acute liver injury in mice. Research Area：Metabolic Disease Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA […]

Benidipine hydrochloride

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Benidipine hydrochloride CAS No. : 91599-74-5 Biological Activity：Benidipine hydrochloride is a dihydropyridine calcium channel blocker for the treatment of high blood pressure (hypertension). Research Area：Cardiovascular Disease Targets：Calcium Channel Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Membrane Transporter/Ion […]