Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Antitumor agent-49 Biological Activity：Antitumor agent-49 (Compound 10) is a Harmine derivative-furoxan hybrids containing NO donor, with antitumor activities. Antitumor agent-49 shows cytotoxic activity against HepG2 cells with an IC50 of 1.79 µM. Antitumor agent-49 produces high levels of NO in vitro. Research Area：Cancer Targets：Others Related Small […]
For research use only. We do not sell to patients. Oleic acid ethanolamine CAS No. : 2272-11-9 Biological Activity：Oleic (9-cis-Octadecenoic) acid ethanolamine consists of oleic acid and ethanolamine. Oleic acid ethanolamine has sclerotherapeutic activity. Oleic acid ethanolamine can cause inflammatory reaction in the intimal endothelium of the vein. Research Area：Inflammation/Immunology|Cardiovascular Disease Targets：Others Related Small Molecules:Immune […]
For research use only. We do not sell to patients. α-Cyano-4-hydroxycinnamic acid CAS No. : 28166-41-8 Biological Activity：α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamate) is a potent and non-competitive inhibitor of monocarboxylate transporters (MCTs). α-Cyano-4-hydroxycinnamic acid inhibits mitochondrial pyruvate transporter with a Ki of 6.3 μM. α-Cyano-4-hydroxycinnamic acid is used as a matrix to facilitate peptide ionization in matrix-assisted […]
For research use only. We do not sell to patients. Valeriandoid F CAS No. : 1427162-60-4 Biological Activity：Valeriandoid F is an iridoid, which potently inhibits NO production with an IC50 value of 0.88 μM. Valeriandoid F has anti-inflammatory and antiproliferative activities. Research Area：Cancer|Inflammation/Immunology Targets：NO Synthase Related Small Molecules:Carboxy-PTIO potassium;Ciwujianoside C3;NOS-IN-3;Regaloside A;Aminopicoline;trans-Isoferulic acid;DETA NONOate;Chondroitin sulfate;3-Bromo-7-nitroindazole;α7 nAchR-JAK2-STAT3 […]
For research use only. We do not sell to patients. D-Glucose-13C,d1-3 Biological Activity：D-Glucose-13C,d1-3 is the deuterium labeled D-Glucose. D-Glucose (Glucose), a monosaccharide, is an important carbohydrate in biology. D-Glucose is a carbohydrate sweetener and critical components of the general metabolism, and serve as critical signaling Research Area：Metabolic Disease|Cancer Targets：Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide […]
For research use only. We do not sell to patients. 6-O-Propynyl-2′-deoxyguanosine CAS No. : 1640051-47-3 Biological Activity：6-O-Propynyl-2′-deoxyguanosine is a click chemistry reagent containing an alkyne group. 6-O-Propynyl-2′-deoxyguanosine can be used for the research of various biochemical. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending […]
For research use only. We do not sell to patients. JAK3/BTK-IN-1 CAS No. : 2674036-91-8 Biological Activity：JAK3/BTK-IN-1 is a potent inhibitor of JAK3/BTK. BTK and JAK3 are two important targets for autoimmune diseases. Simultaneous inhibition of the BTK/JAK3 signalling pathway exhibits synergistic effects. JAK3/BTK-IN-1 has the potential for the research of JAK3 kinase and/or BTK-related […]
For research use only. We do not sell to patients. Abacavir sulfate CAS No. : 188062-50-2 Biological Activity：Abacavir sulfate (Abacavir Hemisulfate) is a competitive, orally active nucleoside reverse transcriptase inhibitor. Abacavir sulfate can inhibits the replication of HIV. Abacavir sulfate shows anticancer activity in prostate cancer cell lines. Abacavir sulfate can trespass the blood-brain-barrier and […]
For research use only. We do not sell to patients. Mosapride-d5 CAS No. : 1246820-66-5 Biological Activity：Mosapride-d5 is the deuterium labeled Mosapride. Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist. Research Area：Neurological Disease Targets：5-HT Receptor Related Small Molecules:F 13714;Nuciferine;Renzapride;LY 344864 racemate;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Tetrahydro-β-carboline;CP-809101;Volinanserin-d4 hydrochloride;Masupirdine free base;BRL-15572 dihydrochloride;LY393558;Brexpiprazole S-oxide […]
For research use only. We do not sell to patients. BI-135585 CAS No. : 1114561-85-1 Biological Activity：BI-135585 is a potent, selective and orally active 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor with an IC50 of 13 nM. BI-135585 exhibits >1000-fold selectivity over other hydroxysteroid dehydrogenases. BI-135585 can be used for type 2 diabetes research[2]. Research Area：Metabolic Disease […]