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Zeteletinib
CAS No. : 2216753-97-6
Biological Activity：Zeteletinib (BOS-172738; DS-5010) is an orally active, selective RET kinase inhibitor with nanomolar potency against RET and >300-fold selectivity against VEGFR2. Zeteletinib shows exquisite potency for the wild type RET, RETV804M/L gatekeeper mutants, and the most common oncogenic RET mutation M918T. Zeteletinib has potent antitumor activity[2][3].
Research Area：Cancer
Targets：RET|PDGFR
Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus;Kinase Inhibitor Library;Protein Tyrosine Kinase Compound Library;Anti-Cancer Compound Library;Clinical Compound Library;Reprogramming Compound Library;Orally Active Compound Library;Anti-Lung Cancer Compound Library;Angiogenesis-Related Compound Library;Anti-Liver Cancer Compound Library ;Anti-Pulmonary Fibrosis Compound Library;
Related Small Molecules:Henatinib;Flumatinib mesylate;IHMT-TRK-284;RET-IN-18;PDGFRα/FLT3-ITD-IN-2;PP58;Chiauranib;ENMD-2076 Tartrate;AZD2932;RET-IN-5;AC710 Mesylate;Tyrosine kinase-IN-1;GSK3179106;Tandutinib;JNJ-10198409;SU4984;Pyrazoloadenine;SU4312;Avapritinib;MELK-8a;trans-Pralsetinib;PF 477736
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