Umbralisib sulfate

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Umbralisib sulfate

CAS No. : 1532533-75-7

Biological Activity:Umbralisib (TGR-1202) sulfate is an orally active, potent and selective dual PI3Kδ and casein kinase-1-ε (CK1ε) inhibitor, with EC50 of 22.2 nM and 6.0 μM, respectively. Umbralisib sulfate exhibits unique immunomodulatory effects on chronic lymphocytic leukemia (CLL) T cells. Umbralisib sulfate can be used for haematological malignancies reseach[2][3][4].

Research Area:Cancer

Targets:Casein Kinase|PI3K

Related Small Molecules:Umbralisib hydrochloride;Topoisomerase I/II inhibitor 3;Rigosertib sodium;Tenalisib R Enantiomer;PI3kδ inhibitor 1;PI3K/VEGFR2-IN-1;1,3-Dicaffeoylquinic acid;PI3Kδ-IN-1;PI-103-d8;PI3Kα-IN-8;4,5,6,7-Tetrabromo-1H-benzimidazole;PI-103 Hydrochloride;IC-87114;PI3K/mTOR Inhibitor-6;PI3K-IN-10;SF2523;TA-01;Ellagic acid;PI3K-IN-29;PI3K/mTOR Inhibitor-1;CK2 inhibitor 3;PI3K-IN-26;GSK-F1;Serabelisib;Amdizalisib;TMCB;Glaucocalyxin A;PI3K/AKT-IN-2;PIK-294

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