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SB-657510
CAS No. : 474960-44-6
Biological Activity：SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The Ki values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells[2].
Research Area：Inflammation/Immunology
Targets：Urotensin Receptor
Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Anti-diabetic Compound Library;Targeted Diversity Library;
Related Small Molecules:Urotensin II, mouse acetate;Palosuran;UFP-803 TFA;[Orn5]-URP;Urotensin II (114-124), human TFA;SB-611812
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