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LP-922761
CAS No. : 1454808-95-7
Biological Activity：LP-922761 is a potent, selective and orally active adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50s of 4.8 nM and 7.6 nM in enzyme and cell assays, respectively. LP-922761 also inhibits BMP-2-inducible protein kinase (BIKE) with an IC50 of 24 nM. LP-922761 exhibits no significant activity at cyclin G-associated kinase (GAK), opioid, adrenergic α2 or GABAa receptors.
Research Area：Neurological Disease
Targets：AAK1
Related Screening Libraries:Bioactive Compound Library Plus;Kinase Inhibitor Library;Neuronal Signaling Compound Library;Orally Active Compound Library;Targeted Diversity Library;Anti-Pulmonary Fibrosis Compound Library;Osteogenesis Compound Library;
Related Small Molecules:DB0614;SGC-AAK1-1;BMS-901715;BMT-090605;BMS-911172;SGC-AAK1-1N;AAK1-IN-2;RSS0680;BMT-124110;AAK1-IN-3 TFA;BMS-986176;LP-935509
Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
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