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BQ-788
CAS No. : 173326-37-9
Biological Activity：BQ-788 is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM.
Research Area：Cardiovascular Disease|Endocrinology
Targets：Endothelin Receptor
Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Clinical Compound Library;Anti-Cardiovascular Disease Compound Library;Endocrinology Compound Library;Ferroptosis Compound Library;Neurotransmitter Receptor Compound Library;Angiogenesis-Related Compound Library;Targeted Diversity Library;Coagulation and Anti-coagulation Compound Library;
Related Small Molecules:[Asn18] Endothelin-1, human;Endothelin-3, human, mouse, rabbit, rat TFA;IRL 2500;Sarafotoxin S6c;Sarafotoxin S6a;ANP (1-30), frog;IRL-1620 TFA;Tezosentan;ACT-373898;Ro 46-2005;Ro 46-8443;[Ala2] Endothelin-3, human;ZD-1611;PD-159020;Aminaftone;Aprocitentan-d4;Endothelin 1 (swine, human);Atrial Natriuretic Peptide (ANP) (1-28), rat;Carperitide acetate;[Ala1,3,11,15]-Endothelin (53-63) (TFA);Sparsentan-d5;BQ-123 TFA
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