Relugolix-d6

For research use only. We do not sell to patients.

Relugolix-d6

Biological Activity:Relugolix-d6 is deuterium labeled Relugolix. Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al[2].

Research Area:Cancer|Endocrinology

Targets:GnRH Receptor

Related Small Molecules:(R)-Elagolix;Linzagolix;[D-Ala6]-LH-RH;Relugolix;Teverelix;Alarelin Acetate;[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide;Kisspeptin 13;opigolix;sGnRH-A;Lecirelin;GnRH-R antagonist 1;Ozarelix;LH-RH (7-10);BAY-298;Acyline;GnRH-I;Lamprey LH-RH I;BAY-784;BAY 1214784;GnRH antagonist 2;[D-Lys6]-LH-RH

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