GSK484 hydrochloride

For research use only. We do not sell to patients.

GSK484 hydrochloride

CAS No. : 1652591-81-5

Biological Activity:GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.

Research Area:Cancer|Inflammation/Immunology|Cardiovascular Disease

Targets:Protein Arginine Deiminase

Related Screening Libraries:Bioactive Compound Library Plus;Epigenetics Compound Library;Immunology/Inflammation Compound Library;Anti-Cancer Compound Library;Anti-Cardiovascular Disease Compound Library;

Related Small Molecules:BMS-P5;BB-Cl-Amidine;D-Cl-amidine;GSK121;Cl-amidine TFA;AFM-30a;PAD2-IN-1;Streptonigrin;PAD-IN-2;GSK199;Acefylline;GSK106

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