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GnRH-R antagonist 1

Biological Activity：GnRH-R antagonist 1 (compound 21a) is an orally safe and membrane-permeable GnRH-R antagonist with high binding affinity (IC₅₀=0.57 nM) and potent in vitro antagonistic activity (IC₅₀=2.18 nM). GnRH-R antagonist 1 can be used in studies of advanced prostate cancer and premature LH peaks preventing.

Research Area：Cancer

Targets：GnRH Receptor

Related Small Molecules:(R)-Elagolix;Linzagolix;Relugolix-d6;[D-Ala6]-LH-RH;Relugolix;Teverelix;Alarelin Acetate;[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide;Kisspeptin 13;opigolix;sGnRH-A;Lecirelin;Ozarelix;LH-RH (7-10);BAY-298;Acyline;GnRH-I;Lamprey LH-RH I;BAY-784;BAY 1214784;GnRH antagonist 2;[D-Lys6]-LH-RH

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