Foropafant

For research use only. We do not sell to patients.

Foropafant

CAS No. : 136468-36-5

Biological Activity:Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor, with a Ki value of 57 pM for [3H]PAF binding, at least 5-fold lower than that of unlabeled PAF itself. Foropafant potently inhibits PAF-induced aggregation of rabbit and human platelets.

Research Area:Cardiovascular Disease

Targets:Platelet-activating Factor Receptor (PAFR)

Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Cardiovascular Disease Compound Library;Orally Active Compound Library;Targeted Diversity Library;Human Metabolite Library;Coagulation and Anti-coagulation Compound Library;

Related Small Molecules:PAF-AN-1;48740 RP;Ro-24-0238;Ro-24-4736;Setipafant;Tulopafant;YM-264;E-​6123;Lexipafant;Homoeriodictyol 7-O-β-D-glucoside;Apafant;CV-6209;(+)-Guaiacin;Modipafant;TCV-309 chloride

Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  |  Oligonucleotides

About Us:

  • MedChemExpress (MCE) offers a wide range of high-quality research chemicals and biochemicals (novel life-science reagents, reference compounds and natural compounds) for scientific use;
  • Structurally and synthetically diverse biologically active compounds;
  •  roduct quality is the key to our success and we take pride in offering only the highest-grade products.;
  • We provide HNMR, LC-MS, HPLC, stability testing and activity assays of our products to clients.;
  • Product identity, quality, purity and activity are assured by our robust quality control programs and procedures.;
  • Structurally and synthetically diverse biologically active compounds;

  • Customized order volume ranging from milligrams to kilograms scale;
  • We provide customer-oriented services. To explore more, please contact us at [email protected]. Our team will gladly assist you.

50K Diversity Library
Top Publications Citing Use of MCE Products
Recombinant Proteins
magnetic-beads