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EST73502
CAS No. : 1838622-25-5
Biological Activity：EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 has antinociceptive activity.
Research Area：Neurological Disease
Targets：Opioid Receptor|Sigma Receptor
Related Small Molecules:ORL1 antagonist 1;Loperamide-d6 N-Oxide;Deltorphin 2 TFA;Nalfurafine;BD1063 dhydrochloride;β-Lipotropin (60-65);GSK1521498 free base;Trimebutine-d5 fumarate;Dynorphin B (1-13) (TFA);Dermorphin Analog;β-Endorphin (6-31), human;Phenyltoloxamine;JTC-801;E1R;Valorphin;Corydaline;TAN-452;Matrine;Naloxonazine dihydrochloride;[Leu5]-Enkephalin;Sec-O-Glucosylhamaudol;DPDPE;CTOP;β-Endorphin, equine;(±)-Vesamicol hydrochloride;Sigma-LIGAND-1
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