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BMS-986202

CAS No. : 1771691-34-9

Biological Activity：BMS-986202 is a potent, selective and orally active Tyk2 inhibitor that binds to Tyk2 JH2 with an IC₅₀ of 0.19 nM and a K_i of 0.02 nM. BMS-986202 is remarkably selective over other kinases including Jak family members. BMS-986202 is also a weak inhibitor of CYP2C19 with an IC₅₀ of 14 μM. BMS-986202 can be used for IL-23-driven acanthosis, anti-CD40-induced colitis, and spontaneous lupus research.

Research Area：Inflammation/Immunology

Targets：JAK|Cytochrome P450

Related Small Molecules:AZ-3;SR9186;JAK3/BTK-IN-1;AMG-208;AT9283;Benzene hexabromide;(E/Z)-Zotiraciclib;CYP1B1-IN-1;CYP2C9/CYP2C19-IN-1;JAK-IN-10;Hypericin;Baricitinib-d3;JAK3-IN-6;Coumermycin A1;Deucravacitinib;Galeterone;Ranitidine;Momelotinib-3,3,5,5-d4;Bergapten;Ginsenoside Rd;SJ10542;Delgocitinib;AS1810722

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