For research use only. We do not sell to patients.
Targefrin
Biological Activity：Targefrin is a potent EphA2-targeting agent, acts as an antagonist. Targefrin binds EphA2-LBD with 21 nM dissociation constant and an IC50 value of 10.8 nM. Targefrin induces cellular receptor internalization and degradation in several pancreatic cancer cell lines.
Research Area：Cancer
Targets：Ephrin Receptor
Related Small Molecules:LDN-211904 oxalate;KYL peptide;UniPR129;EphA2 agonist 2;ALW-II-41-27;JI-101;Eph inhibitor 2;UniPR505;ML786 dihydrochloride;NVP-BHG712;Tesevatinib;BT5528;123C4;EphA2 agonist 1
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Structurally and synthetically diverse biologically active compounds；
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