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RP101075

CAS No. : 1306760-73-5

Biological Activity：RP101075, an active metabolite of Ozanimod, is a potent, orally active S1PR (sphingosine-1-phosphate receptor 1) agonist, with an EC₅₀ of 0.27 nM. RP101075 displays >100-fold selectivity over S1PR5 (EC₅₀=5.9 nM) and >10000-fold over S1PR 2, 3, and 4. RP101075 displays superior cardiovascular safety profile.

Research Area：Inflammation/Immunology

Targets：Drug Metabolite|LPL Receptor

Related Small Molecules:Nicotinamide N-oxide;GSK2018682;4-Hydroxyphenylbutazone;Ampyrone;Resveratrol-3-O-sulfate sodium;Sonidegib metabolite M48;Isonicotinic acid;Ozanimod hydrochloride;Cycloguanil hydrochloride;BMS-986020 sodium;S1p receptor agonist 2;ONO-9780307;Siponimod hemifumarate;Hydroxytanshinone IIA;S1P2 antagonist 1;S1P1 agonist III;Endoxifen;Ceralifimod

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