Rimegepant

For research use only. We do not sell to patients.

Rimegepant

CAS No. : 1289023-67-1

Biological Activity:Rimegepant (BMS-927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki of 0.027 nM and an IC50 of 0.14 nM for hCGRP receptor.

Research Area:Neurological Disease

Targets:CGRP Receptor

Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;FDA-Approved Drug Library;Drug Repurposing Compound Library;Orally Active Compound Library;FDA Approved & Pharmacopeial Drug Library;Drug-Induced Liver Injury (DILI) Compound Library;Targeted Diversity Library;Human Metabolite Library;

Related Small Molecules:Vazegepant hydrochloride;Adrenomedullin (16-31), human;MK-3207 Hydrochloride;α-CGRP, rat;Cagrilintide acetate;HTL22562;SUN B8155;Adrenomedullin (11-50), rat;Rat CGRP-(8-37);Atogepant;β-CGRP, human TFA;Calcitonin (salmon);Calcitonin (human);α-CGRP(human);Galcanezumab;Olcegepant;Calcitonin Gene Related Peptide (CGRP) II, rat;Ubrogepant;PHM-27 (human);Adrenomedullin (1-50), rat;CGRP antagonist 1;Telcagepant;HCGRP-(8-37)

Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  |  Oligonucleotides

About Us:

  • MedChemExpress (MCE) offers a wide range of high-quality research chemicals and biochemicals (novel life-science reagents, reference compounds and natural compounds) for scientific use;
  • Structurally and synthetically diverse biologically active compounds;
  •  roduct quality is the key to our success and we take pride in offering only the highest-grade products.;
  • We provide HNMR, LC-MS, HPLC, stability testing and activity assays of our products to clients.;
  • Product identity, quality, purity and activity are assured by our robust quality control programs and procedures.;
  • Structurally and synthetically diverse biologically active compounds;

  • Customized order volume ranging from milligrams to kilograms scale;
  • We provide customer-oriented services. To explore more, please contact us at [email protected]. Our team will gladly assist you.

50K Diversity Library
Top Publications Citing Use of MCE Products
Recombinant Proteins
magnetic-beads