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PROTAC CDK2/9 Degrader-1

CAS No. : 2408641-24-5

Biological Activity：PROTAC CDK2/9 Degrader-1 (Compound F3) is a potent dual degrader for CDK2 (DC₅₀=62 nM) and CDK9 (DC₅₀=33 nM). PROTAC CDK2/9 Degrader-1 suppresses prostate cancer PC-3 cell proliferation (IC₅₀=0.12 µM) by effectively blocking the cell cycle in S and G2/M phases. PROTAC CDK2/9 Degrader-1 is a PROTAC by tethering CDK inhibitor with Cereblon ligand.

Research Area：Cancer

Targets：CDK|PROTACs

Related Screening Libraries:Bioactive Compound Library Plus;

Related Small Molecules:PROTAC Sirt2 Degrader-1;DB0614;Dinaciclib;SNS-032;CC-671;PROTAC VEGFR-2 degrader-2;(E/Z)-Zotiraciclib;dTAGV-1-NEG;CCT367766 formic;CDK1-IN-4;CCT-251921;BS-181;Samuraciclib hydrochloride hydrate;T025;HDAC6 degrader-1;Flavopiridol;CDK8-IN-3;PROTAC Axl Degrader 2;PhosTAC7;CDK9-IN-12;MS98;FLT3/CDK4-IN-1;GFB-12811;GSK 3 Inhibitor IX;JPS014;Eciruciclib;PROTAC PARP1 degrader;MD-224;CDK-IN-6

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